Assay Detail
Functional
CHEMBL2363569
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SANGER: Inhibition of human OCUB-M cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OCUB-M |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.76 | 9.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.35 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.22 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.99 |
| CHEMBL1256459 | TORIN1 | — | 1 | 8.71 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.36 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.35 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.18 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.12 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.00 |
| CHEMBL514499 | GW843682X | — | 1 | 7.91 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.82 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.74 |
| CHEMBL379300 | A-443654 | — | 1 | 7.59 |
| CHEMBL64925 | MG-132 | — | 2 | 7.43 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.42 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.40 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 7.35 |
| CHEMBL300389 | — | — | 1 | 7.28 |
| CHEMBL554 | LAPATINIB | 4.0 | 1 | 7.24 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.08 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.99 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 6.77 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.65 |
| CHEMBL217354 | — | — | 1 | 6.62 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.46 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 6.33 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.15 |
| CHEMBL2165191 | AZD-6482 | 2.0 | 2 | 6.14 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 6.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.4469 | nM | 9.35 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.5967 | nM | 9.22 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.025 | nM | 8.99 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 1.94 | nM | 8.71 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 4.379 | nM | 8.36 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 4.433 | nM | 8.35 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 6.617 | nM | 8.18 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 7.561 | nM | 8.12 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 10.03 | nM | 8.00 |
| CHEMBL514499 | GW843682X | IC50 | = | 12.21 | nM | 7.91 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 15.15 | nM | 7.82 |
| CHEMBL513909 | BI-2536 | IC50 | = | 18.26 | nM | 7.74 |
| CHEMBL379300 | A-443654 | IC50 | = | 25.73 | nM | 7.59 |
| CHEMBL64925 | MG-132 | IC50 | = | 37.37 | nM | 7.43 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 38.13 | nM | 7.42 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 39.61 | nM | 7.40 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 44.55 | nM | 7.35 |
| CHEMBL300389 | — | IC50 | = | 52.55 | nM | 7.28 |
| CHEMBL554 | LAPATINIB | IC50 | = | 57.4 | nM | 7.24 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 82.41 | nM | 7.08 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 102.98 | nM | 6.99 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 169.83 | nM | 6.77 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 195.45 | nM | 6.71 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 224.88 | nM | 6.65 |
| CHEMBL217354 | — | IC50 | = | 242.77 | nM | 6.62 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 350.38 | nM | 6.46 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 471.64 | nM | 6.33 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 709.66 | nM | 6.15 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 727.88 | nM | 6.14 |
| CHEMBL2363137 | — | IC50 | = | 810.3 | nM | 6.09 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 816.89 | nM | 6.09 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 805.64 | nM | 6.09 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 826.75 | nM | 6.08 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 865.23 | nM | 6.06 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 1021.91 | nM | 5.99 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 1044.12 | nM | 5.98 |
| CHEMBL191384 | — | IC50 | = | 1081.07 | nM | 5.97 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 1082.94 | nM | 5.96 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1214.89 | nM | 5.92 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1361.43 | nM | 5.87 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1359.15 | nM | 5.87 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1553.73 | nM | 5.81 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1583.14 | nM | 5.80 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1813.57 | nM | 5.74 |
| CHEMBL1643959 | — | IC50 | = | 2097.0 | nM | 5.68 |
| CHEMBL202721 | — | IC50 | = | 2250.52 | nM | 5.65 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 2342.86 | nM | 5.63 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 2788.61 | nM | 5.55 |
| CHEMBL585951 | — | IC50 | = | 3034.4 | nM | 5.52 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 3313.68 | nM | 5.48 |