Assay Detail
Functional
CHEMBL2363578
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human OVCAR-5 cell growth in a cell viability assay.
98
Total Activities
97
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OVCAR-5 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 98 | 5.90 | 9.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.40 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.74 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.70 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.55 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 8.11 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.87 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.74 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.46 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.45 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.36 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.96 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.93 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.91 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.86 |
| CHEMBL585951 | — | — | 1 | 6.74 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.66 |
| CHEMBL3349342 | — | — | 1 | 6.63 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.51 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.51 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.37 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.35 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.31 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.30 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.30 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.24 |
| CHEMBL217354 | — | — | 1 | 6.24 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.16 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.05 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.03 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.95 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.3985 | nM | 9.40 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1.835 | nM | 8.74 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.994 | nM | 8.70 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 2.84 | nM | 8.55 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 7.823 | nM | 8.11 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 13.6 | nM | 7.87 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 18.12 | nM | 7.74 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 34.8 | nM | 7.46 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 35.47 | nM | 7.45 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 43.33 | nM | 7.36 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 110.16 | nM | 6.96 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 116.81 | nM | 6.93 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 123.69 | nM | 6.91 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 138.94 | nM | 6.86 |
| CHEMBL585951 | — | IC50 | = | 181.32 | nM | 6.74 |
| CHEMBL803 | CYTARABINE | IC50 | = | 219.63 | nM | 6.66 |
| CHEMBL3349342 | — | IC50 | = | 234.19 | nM | 6.63 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 305.77 | nM | 6.51 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 311.06 | nM | 6.51 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 429.33 | nM | 6.37 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 445.47 | nM | 6.35 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 487.11 | nM | 6.31 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 503.56 | nM | 6.30 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 502.07 | nM | 6.30 |
| CHEMBL217354 | — | IC50 | = | 575.72 | nM | 6.24 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 576.11 | nM | 6.24 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 691.67 | nM | 6.16 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 900.1 | nM | 6.05 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 940.17 | nM | 6.03 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1123.89 | nM | 5.95 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1537.48 | nM | 5.81 |
| CHEMBL105442 | CI-1040 | IC50 | = | 1776.87 | nM | 5.75 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 1906.75 | nM | 5.72 |
| CHEMBL577784 | BX-795 | IC50 | = | 2277.34 | nM | 5.64 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 3363.52 | nM | 5.47 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 4023.89 | nM | 5.39 |
| CHEMBL176544 | — | IC50 | = | 4399.53 | nM | 5.36 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 4748.99 | nM | 5.32 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 4812.26 | nM | 5.32 |
| CHEMBL1190711 | — | IC50 | = | 7411.32 | nM | 5.13 |
| CHEMBL573107 | — | IC50 | = | 7823.29 | nM | 5.11 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 8776.25 | nM | 5.06 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 10243.33 | nM | 4.99 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 10642.93 | nM | 4.97 |
| CHEMBL477989 | SB590885 | IC50 | = | 12897.53 | nM | 4.89 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 13159.32 | nM | 4.88 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 14668.74 | nM | 4.83 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 21003.39 | nM | 4.68 |
| CHEMBL2363137 | — | IC50 | = | 23559.24 | nM | 4.63 |
| CHEMBL393929 | — | IC50 | = | 24103.98 | nM | 4.62 |