Assay Detail
Functional
CHEMBL2363580
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SANGER: Inhibition of human P12-ICHIKAWA cell growth in a cell viability assay.
90
Total Activities
90
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | P12-Ichikawa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 90 | 6.09 | 9.99 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.99 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.13 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.77 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.39 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.32 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 8.26 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.96 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.89 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.82 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.61 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.60 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 7.58 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.38 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 7.37 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.31 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.21 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.13 |
| CHEMBL443684 | NAVITOCLAX | 3.0 | 1 | 7.11 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.07 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 7.02 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.93 |
| CHEMBL202721 | — | — | 1 | 6.65 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.50 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 6.48 |
| CHEMBL379975 | — | — | 1 | 6.32 |
| CHEMBL512504 | — | — | 1 | 6.31 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.30 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.22 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 6.21 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.99 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.1016 | nM | 9.99 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.7452 | nM | 9.13 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.704 | nM | 8.77 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 4.044 | nM | 8.39 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 4.787 | nM | 8.32 |
| CHEMBL803 | CYTARABINE | IC50 | = | 5.537 | nM | 8.26 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 11.02 | nM | 7.96 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 13.01 | nM | 7.89 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 15.1 | nM | 7.82 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 24.54 | nM | 7.61 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 25.15 | nM | 7.60 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 26.18 | nM | 7.58 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 41.3 | nM | 7.38 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 43.16 | nM | 7.37 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 49.27 | nM | 7.31 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 62.27 | nM | 7.21 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 73.49 | nM | 7.13 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 77.78 | nM | 7.11 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 84.7 | nM | 7.07 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 96.04 | nM | 7.02 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 116.2 | nM | 6.93 |
| CHEMBL202721 | — | IC50 | = | 224.41 | nM | 6.65 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 316.79 | nM | 6.50 |
| CHEMBL939 | GEFITINIB | IC50 | = | 328.06 | nM | 6.48 |
| CHEMBL379975 | — | IC50 | = | 482.02 | nM | 6.32 |
| CHEMBL512504 | — | IC50 | = | 488.62 | nM | 6.31 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 498.25 | nM | 6.30 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 596.51 | nM | 6.22 |
| CHEMBL105442 | CI-1040 | IC50 | = | 612.21 | nM | 6.21 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1034.06 | nM | 5.99 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1158.99 | nM | 5.94 |
| CHEMBL577784 | BX-795 | IC50 | = | 1181.71 | nM | 5.93 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1388.36 | nM | 5.86 |
| CHEMBL3349342 | — | IC50 | = | 1776.46 | nM | 5.75 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 2040.15 | nM | 5.69 |
| CHEMBL573107 | — | IC50 | = | 2525.59 | nM | 5.60 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 2820.46 | nM | 5.55 |
| CHEMBL477989 | SB590885 | IC50 | = | 3439.95 | nM | 5.46 |
| CHEMBL585951 | — | IC50 | = | 3810.09 | nM | 5.42 |
| CHEMBL1190711 | — | IC50 | = | 4366.12 | nM | 5.36 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 5401.0 | nM | 5.27 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 5545.75 | nM | 5.26 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 7455.23 | nM | 5.13 |
| CHEMBL259181 | — | IC50 | = | 7932.7 | nM | 5.10 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 8789.4 | nM | 5.06 |
| CHEMBL221137 | EMBELIN | IC50 | = | 9449.58 | nM | 5.03 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 9282.82 | nM | 5.03 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 10416.02 | nM | 4.98 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 11109.55 | nM | 4.95 |
| CHEMBL189584 | PD-173074 | IC50 | = | 12384.54 | nM | 4.91 |