Assay Detail
Functional
CHEMBL2363584
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SANGER: Inhibition of human PANC-03-27 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PANC-03-27 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.91 | 10.04 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 10.04 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.88 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.81 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.45 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.26 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.23 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.15 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.93 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.55 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.40 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.01 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.99 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.84 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.79 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.78 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.78 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.70 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.60 |
| CHEMBL585951 | — | — | 1 | 6.57 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.50 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.47 |
| CHEMBL217354 | — | — | 1 | 6.32 |
| CHEMBL591429 | PAC-1 | 1.0 | 1 | 6.12 |
| CHEMBL3349342 | — | — | 1 | 6.11 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.05 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.99 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 5.93 |
| CHEMBL379975 | — | — | 1 | 5.92 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.09108 | nM | 10.04 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.132 | nM | 9.88 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.537 | nM | 8.81 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 3.513 | nM | 8.45 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 5.472 | nM | 8.26 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 5.948 | nM | 8.23 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 7.103 | nM | 8.15 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 11.62 | nM | 7.93 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 28.16 | nM | 7.55 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 39.91 | nM | 7.40 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 76.25 | nM | 7.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 96.71 | nM | 7.01 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 102.86 | nM | 6.99 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 142.88 | nM | 6.84 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 160.2 | nM | 6.79 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 167.16 | nM | 6.78 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 167.4 | nM | 6.78 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 200.85 | nM | 6.70 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 250.74 | nM | 6.60 |
| CHEMBL585951 | — | IC50 | = | 270.89 | nM | 6.57 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 316.39 | nM | 6.50 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 341.97 | nM | 6.47 |
| CHEMBL217354 | — | IC50 | = | 474.14 | nM | 6.32 |
| CHEMBL591429 | PAC-1 | IC50 | = | 759.67 | nM | 6.12 |
| CHEMBL3349342 | — | IC50 | = | 768.35 | nM | 6.11 |
| CHEMBL803 | CYTARABINE | IC50 | = | 896.62 | nM | 6.05 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1031.41 | nM | 5.99 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1170.05 | nM | 5.93 |
| CHEMBL379975 | — | IC50 | = | 1208.34 | nM | 5.92 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 1514.08 | nM | 5.82 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1636.9 | nM | 5.79 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1701.39 | nM | 5.77 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 1842.92 | nM | 5.73 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 2166.31 | nM | 5.66 |
| CHEMBL191384 | — | IC50 | = | 2897.36 | nM | 5.54 |
| CHEMBL105442 | CI-1040 | IC50 | = | 3350.45 | nM | 5.47 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 3819.16 | nM | 5.42 |
| CHEMBL577784 | BX-795 | IC50 | = | 4214.01 | nM | 5.38 |
| CHEMBL573107 | — | IC50 | = | 4300.83 | nM | 5.37 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4399.2 | nM | 5.36 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 4539.29 | nM | 5.34 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 4999.62 | nM | 5.30 |
| CHEMBL1190711 | — | IC50 | = | 5557.98 | nM | 5.25 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 5725.58 | nM | 5.24 |
| CHEMBL2363137 | — | IC50 | = | 6379.09 | nM | 5.20 |
| CHEMBL202721 | — | IC50 | = | 6427.61 | nM | 5.19 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 7927.15 | nM | 5.10 |
| CHEMBL259181 | — | IC50 | = | 7890.92 | nM | 5.10 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 8369.2 | nM | 5.08 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 8487.2 | nM | 5.07 |