Assay Detail
Functional
CHEMBL2363620
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human SAS cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SAS |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.45 | 8.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.91 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.87 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.69 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.65 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.55 |
| CHEMBL217354 | — | — | 1 | 7.48 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.04 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.97 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.97 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.94 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.90 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.56 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 6.46 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.37 |
| CHEMBL1173655 | AFATINIB | 4.0 | 1 | 6.32 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.21 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.18 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.07 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.02 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 5.98 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 5.90 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 5.90 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.82 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 5.81 |
| CHEMBL585951 | — | — | 1 | 5.71 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.66 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.56 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 5.52 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 5.49 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 5.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.241 | nM | 8.91 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.336 | nM | 8.87 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 20.5 | nM | 7.69 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 22.5 | nM | 7.65 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 28.13 | nM | 7.55 |
| CHEMBL217354 | — | IC50 | = | 33.18 | nM | 7.48 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 92.15 | nM | 7.04 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 106.42 | nM | 6.97 |
| CHEMBL803 | CYTARABINE | IC50 | = | 107.57 | nM | 6.97 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 114.45 | nM | 6.94 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 126.9 | nM | 6.90 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 273.08 | nM | 6.56 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 344.06 | nM | 6.46 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 424.6 | nM | 6.37 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 483.98 | nM | 6.32 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 614.65 | nM | 6.21 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 652.67 | nM | 6.18 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 853.74 | nM | 6.07 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 957.68 | nM | 6.02 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 1040.81 | nM | 5.98 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 1266.72 | nM | 5.90 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 1267.2 | nM | 5.90 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1516.22 | nM | 5.82 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 1547.74 | nM | 5.81 |
| CHEMBL585951 | — | IC50 | = | 1943.36 | nM | 5.71 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 2203.74 | nM | 5.66 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 2765.0 | nM | 5.56 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 2994.15 | nM | 5.52 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 3261.45 | nM | 5.49 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 3937.81 | nM | 5.41 |
| CHEMBL3349342 | — | IC50 | = | 3942.98 | nM | 5.40 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 4391.25 | nM | 5.36 |
| CHEMBL259181 | — | IC50 | = | 4800.7 | nM | 5.32 |
| CHEMBL379975 | — | IC50 | = | 4925.82 | nM | 5.31 |
| CHEMBL399530 | — | IC50 | = | 5242.57 | nM | 5.28 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 5873.8 | nM | 5.23 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 9255.81 | nM | 5.03 |
| CHEMBL573107 | — | IC50 | = | 9584.55 | nM | 5.02 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 9903.34 | nM | 5.00 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 10248.02 | nM | 4.99 |
| CHEMBL191384 | — | IC50 | = | 12063.05 | nM | 4.92 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 12859.98 | nM | 4.89 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 13308.09 | nM | 4.88 |
| CHEMBL105442 | CI-1040 | IC50 | = | 15937.34 | nM | 4.80 |
| CHEMBL1186585 | — | IC50 | = | 15862.46 | nM | 4.80 |
| CHEMBL221137 | EMBELIN | IC50 | = | 16808.94 | nM | 4.77 |
| CHEMBL1090771 | AVAGACESTAT | IC50 | = | 17781.24 | nM | 4.75 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 18542.57 | nM | 4.73 |
| CHEMBL2134202 | — | IC50 | = | 18645.45 | nM | 4.73 |
| CHEMBL135561 | — | IC50 | = | 22632.34 | nM | 4.64 |