Assay Detail
Functional
CHEMBL2363642
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SANGER: Inhibition of human SK-LMS-1 cell growth in a cell viability assay.
118
Total Activities
116
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SK-LMS-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 118 | 5.83 | 9.65 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.65 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.24 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.19 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.07 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.84 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 8.60 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.40 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.34 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.85 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.27 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.24 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.23 |
| CHEMBL514499 | GW843682X | — | 1 | 7.13 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.96 |
| CHEMBL300389 | — | — | 1 | 6.87 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 6.74 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.74 |
| CHEMBL64925 | MG-132 | — | 2 | 6.71 |
| CHEMBL217354 | — | — | 1 | 6.57 |
| CHEMBL379300 | A-443654 | — | 1 | 6.56 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.50 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.45 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.36 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.36 |
| CHEMBL585951 | — | — | 1 | 6.34 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.26 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.18 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.11 |
| CHEMBL450786 | PHA-665752 | — | 1 | 6.05 |
| CHEMBL509032 | TAE-684 | — | 1 | 5.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.2255 | nM | 9.65 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.5776 | nM | 9.24 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.646 | nM | 9.19 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.854 | nM | 9.07 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 1.461 | nM | 8.84 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 2.495 | nM | 8.60 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 4.006 | nM | 8.40 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 4.575 | nM | 8.34 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 14.13 | nM | 7.85 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 53.22 | nM | 7.27 |
| CHEMBL513909 | BI-2536 | IC50 | = | 58.05 | nM | 7.24 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 58.6 | nM | 7.23 |
| CHEMBL514499 | GW843682X | IC50 | = | 73.39 | nM | 7.13 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 108.41 | nM | 6.96 |
| CHEMBL300389 | — | IC50 | = | 134.77 | nM | 6.87 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 180.87 | nM | 6.74 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 184.09 | nM | 6.74 |
| CHEMBL64925 | MG-132 | IC50 | = | 193.03 | nM | 6.71 |
| CHEMBL217354 | — | IC50 | = | 271.51 | nM | 6.57 |
| CHEMBL379300 | A-443654 | IC50 | = | 276.37 | nM | 6.56 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 314.29 | nM | 6.50 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 353.35 | nM | 6.45 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 436.61 | nM | 6.36 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 439.29 | nM | 6.36 |
| CHEMBL585951 | — | IC50 | = | 452.54 | nM | 6.34 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 552.8 | nM | 6.26 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 664.7 | nM | 6.18 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 773.09 | nM | 6.11 |
| CHEMBL450786 | PHA-665752 | IC50 | = | 898.46 | nM | 6.05 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1159.74 | nM | 5.94 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 1222.12 | nM | 5.91 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1396.9 | nM | 5.86 |
| CHEMBL515416 | — | IC50 | = | 1398.57 | nM | 5.85 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 1768.67 | nM | 5.75 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 2657.61 | nM | 5.58 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 2641.28 | nM | 5.58 |
| CHEMBL259181 | — | IC50 | = | 2940.87 | nM | 5.53 |
| CHEMBL2363137 | — | IC50 | = | 3097.02 | nM | 5.51 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 3070.71 | nM | 5.51 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 3118.86 | nM | 5.51 |
| CHEMBL535 | SUNITINIB | IC50 | = | 3833.38 | nM | 5.42 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4615.97 | nM | 5.34 |
| CHEMBL401930 | — | IC50 | = | 4813.91 | nM | 5.32 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 5382.55 | nM | 5.27 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5642.74 | nM | 5.25 |
| CHEMBL399530 | — | IC50 | = | 6839.79 | nM | 5.17 |
| CHEMBL191384 | — | IC50 | = | 7384.56 | nM | 5.13 |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 7624.74 | nM | 5.12 |
| CHEMBL258844 | — | IC50 | = | 8764.52 | nM | 5.06 |
| CHEMBL2134202 | — | IC50 | = | 9013.02 | nM | 5.04 |