Assay Detail
Functional
CHEMBL2363692
Review assay metadata, readout intent, target linkage, and publication context from the same page.
SANGER: Inhibition of human SW872 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SW872 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.82 | 9.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 9.17 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.12 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.11 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 9.07 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.00 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.25 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.24 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 7.73 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.65 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.62 |
| CHEMBL300389 | — | — | 1 | 7.58 |
| CHEMBL514499 | GW843682X | — | 1 | 7.56 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 7.55 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.49 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.38 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.38 |
| CHEMBL217354 | — | — | 1 | 7.23 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.19 |
| CHEMBL2144069 | — | — | 1 | 7.02 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.92 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 6.79 |
| CHEMBL379300 | A-443654 | — | 1 | 6.59 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.59 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.57 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.43 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.35 |
| CHEMBL197603 | — | — | 1 | 6.34 |
| CHEMBL585951 | — | — | 1 | 6.27 |
| CHEMBL509032 | TAE-684 | — | 1 | 6.25 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL105 | MITOMYCIN | IC50 | = | 0.676 | nM | 9.17 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.7647 | nM | 9.12 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7737 | nM | 9.11 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 0.8464 | nM | 9.07 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.9964 | nM | 9.00 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 5.65 | nM | 8.25 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 5.776 | nM | 8.24 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 18.67 | nM | 7.73 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 22.47 | nM | 7.65 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 24.16 | nM | 7.62 |
| CHEMBL300389 | — | IC50 | = | 26.6 | nM | 7.58 |
| CHEMBL514499 | GW843682X | IC50 | = | 27.75 | nM | 7.56 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 27.99 | nM | 7.55 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 32.17 | nM | 7.49 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 42.1 | nM | 7.38 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 41.61 | nM | 7.38 |
| CHEMBL217354 | — | IC50 | = | 58.9 | nM | 7.23 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 64.57 | nM | 7.19 |
| CHEMBL2144069 | — | IC50 | = | 96.48 | nM | 7.02 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 120.81 | nM | 6.92 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 160.42 | nM | 6.79 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 255.22 | nM | 6.59 |
| CHEMBL379300 | A-443654 | IC50 | = | 255.39 | nM | 6.59 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 269.85 | nM | 6.57 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 367.48 | nM | 6.43 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 446.57 | nM | 6.35 |
| CHEMBL197603 | — | IC50 | = | 452.21 | nM | 6.34 |
| CHEMBL585951 | — | IC50 | = | 538.89 | nM | 6.27 |
| CHEMBL509032 | TAE-684 | IC50 | = | 567.24 | nM | 6.25 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 607.63 | nM | 6.22 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 640.4 | nM | 6.19 |
| CHEMBL64925 | MG-132 | IC50 | = | 657.29 | nM | 6.18 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 727.89 | nM | 6.14 |
| CHEMBL3349342 | — | IC50 | = | 774.23 | nM | 6.11 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 794.57 | nM | 6.10 |
| CHEMBL213100 | — | IC50 | = | 864.58 | nM | 6.06 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 886.56 | nM | 6.05 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 944.59 | nM | 6.03 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 997.75 | nM | 6.00 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 993.24 | nM | 6.00 |
| CHEMBL1190711 | — | IC50 | = | 1176.05 | nM | 5.93 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 1268.55 | nM | 5.90 |
| CHEMBL191384 | — | IC50 | = | 1322.18 | nM | 5.88 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1385.55 | nM | 5.86 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1451.0 | nM | 5.84 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1813.95 | nM | 5.74 |
| CHEMBL401930 | — | IC50 | = | 1980.52 | nM | 5.70 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1983.3 | nM | 5.70 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 2185.07 | nM | 5.66 |
| CHEMBL64925 | MG-132 | IC50 | = | 2600.22 | nM | 5.58 |