Assay Detail
Functional
CHEMBL2363696
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SANGER: Inhibition of human SW962 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SW 962 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.62 | 8.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.98 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.53 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.28 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.18 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.16 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.81 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.71 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.69 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.63 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.57 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.55 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.54 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.40 |
| CHEMBL514499 | GW843682X | — | 1 | 7.38 |
| CHEMBL300389 | — | — | 1 | 7.35 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.28 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.18 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.16 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.11 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.95 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.95 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.81 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.80 |
| CHEMBL379300 | A-443654 | — | 1 | 6.59 |
| CHEMBL217354 | — | — | 1 | 6.42 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.33 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.25 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 6.13 |
| CHEMBL189584 | PD-173074 | — | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.036 | nM | 8.98 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 2.929 | nM | 8.53 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 5.208 | nM | 8.28 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 6.623 | nM | 8.18 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 6.848 | nM | 8.16 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 15.59 | nM | 7.81 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 19.39 | nM | 7.71 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 20.51 | nM | 7.69 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 23.36 | nM | 7.63 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 26.76 | nM | 7.57 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 27.83 | nM | 7.55 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 28.52 | nM | 7.54 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 39.45 | nM | 7.40 |
| CHEMBL514499 | GW843682X | IC50 | = | 42.17 | nM | 7.38 |
| CHEMBL300389 | — | IC50 | = | 45.1 | nM | 7.35 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 52.41 | nM | 7.28 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 57.63 | nM | 7.24 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 65.69 | nM | 7.18 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 69.95 | nM | 7.16 |
| CHEMBL513909 | BI-2536 | IC50 | = | 78.39 | nM | 7.11 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 112.92 | nM | 6.95 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 111.28 | nM | 6.95 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 153.92 | nM | 6.81 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 157.55 | nM | 6.80 |
| CHEMBL379300 | A-443654 | IC50 | = | 254.68 | nM | 6.59 |
| CHEMBL217354 | — | IC50 | = | 377.91 | nM | 6.42 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 471.9 | nM | 6.33 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 568.3 | nM | 6.25 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 748.44 | nM | 6.13 |
| CHEMBL189584 | PD-173074 | IC50 | = | 789.88 | nM | 6.10 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 808.63 | nM | 6.09 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 969.11 | nM | 6.01 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1084.87 | nM | 5.96 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1138.11 | nM | 5.94 |
| CHEMBL401930 | — | IC50 | = | 1200.86 | nM | 5.92 |
| CHEMBL213100 | — | IC50 | = | 1337.42 | nM | 5.87 |
| CHEMBL3349342 | — | IC50 | = | 1499.27 | nM | 5.82 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1504.79 | nM | 5.82 |
| CHEMBL509032 | TAE-684 | IC50 | = | 1561.3 | nM | 5.81 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1954.52 | nM | 5.71 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 2040.59 | nM | 5.69 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2153.91 | nM | 5.67 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 2171.78 | nM | 5.66 |
| CHEMBL577784 | BX-795 | IC50 | = | 2337.57 | nM | 5.63 |
| CHEMBL188678 | — | IC50 | = | 3203.52 | nM | 5.49 |
| CHEMBL515416 | — | IC50 | = | 3660.99 | nM | 5.44 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 3726.36 | nM | 5.43 |
| CHEMBL803 | CYTARABINE | IC50 | = | 3739.62 | nM | 5.43 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 4364.27 | nM | 5.36 |
| CHEMBL2363137 | — | IC50 | = | 4681.29 | nM | 5.33 |