Assay Detail
Functional
CHEMBL2363703
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SANGER: Inhibition of human T98G cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T98G |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.53 | 9.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.13 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.93 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.94 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.72 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 7.70 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.58 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.57 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.53 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.46 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.39 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.13 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.72 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 6.71 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.61 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.59 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.49 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.28 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.27 |
| CHEMBL585951 | — | — | 1 | 6.25 |
| CHEMBL217354 | — | — | 1 | 6.22 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 5.99 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.97 |
| CHEMBL393929 | — | — | 1 | 5.86 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 5.76 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 5.70 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 5.70 |
| CHEMBL577784 | BX-795 | — | 1 | 5.62 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.55 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 5.52 |
| CHEMBL573107 | — | — | 1 | 5.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.7406 | nM | 9.13 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.17 | nM | 8.93 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 11.4 | nM | 7.94 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 18.91 | nM | 7.72 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 19.96 | nM | 7.70 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 26.17 | nM | 7.58 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 27.15 | nM | 7.57 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 29.88 | nM | 7.53 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 34.31 | nM | 7.46 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 41.03 | nM | 7.39 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 74.21 | nM | 7.13 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 189.95 | nM | 6.72 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 193.18 | nM | 6.71 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 245.68 | nM | 6.61 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 257.16 | nM | 6.59 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 327.36 | nM | 6.49 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 523.75 | nM | 6.28 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 539.48 | nM | 6.27 |
| CHEMBL585951 | — | IC50 | = | 567.01 | nM | 6.25 |
| CHEMBL217354 | — | IC50 | = | 606.12 | nM | 6.22 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1013.64 | nM | 5.99 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1082.08 | nM | 5.97 |
| CHEMBL393929 | — | IC50 | = | 1368.12 | nM | 5.86 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1718.11 | nM | 5.76 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 1990.06 | nM | 5.70 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 2006.66 | nM | 5.70 |
| CHEMBL577784 | BX-795 | IC50 | = | 2388.57 | nM | 5.62 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 2804.01 | nM | 5.55 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 3013.13 | nM | 5.52 |
| CHEMBL573107 | — | IC50 | = | 3282.16 | nM | 5.48 |
| CHEMBL202721 | — | IC50 | = | 3950.05 | nM | 5.40 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 4221.57 | nM | 5.38 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 5065.08 | nM | 5.29 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 5529.55 | nM | 5.26 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 5796.35 | nM | 5.24 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 7300.92 | nM | 5.14 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 8180.67 | nM | 5.09 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 8434.4 | nM | 5.07 |
| CHEMBL105442 | CI-1040 | IC50 | = | 8998.46 | nM | 5.05 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 8815.81 | nM | 5.05 |
| CHEMBL1289926 | AXITINIB | IC50 | = | 9902.03 | nM | 5.00 |
| CHEMBL2363137 | — | IC50 | = | 10627.88 | nM | 4.97 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 11796.57 | nM | 4.93 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 12845.93 | nM | 4.89 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 13471.74 | nM | 4.87 |
| CHEMBL191384 | — | IC50 | = | 14009.45 | nM | 4.85 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 16246.93 | nM | 4.79 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 18515.66 | nM | 4.73 |
| CHEMBL221137 | EMBELIN | IC50 | = | 19646.91 | nM | 4.71 |
| CHEMBL102714 | SB-216763 | IC50 | = | 23300.92 | nM | 4.63 |