Assay Detail
Functional
CHEMBL2363714
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SANGER: Inhibition of human 769-P cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | 769-P |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.74 | 9.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 9.91 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.17 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 8.15 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.01 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.98 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.97 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.77 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.68 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.60 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.59 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.49 |
| CHEMBL34259 | METHOTREXATE | 4.0 | 1 | 7.34 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.13 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.92 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.91 |
| CHEMBL217354 | — | — | 1 | 6.86 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 6.80 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.67 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.65 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.64 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.40 |
| CHEMBL585951 | — | — | 1 | 6.27 |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | 6.23 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.16 |
| CHEMBL1190711 | — | — | 1 | 6.01 |
| CHEMBL379975 | — | — | 1 | 5.99 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.92 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 5.89 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 5.79 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL888 | GEMCITABINE | IC50 | = | 0.1231 | nM | 9.91 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7534 | nM | 9.12 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 6.778 | nM | 8.17 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 7.112 | nM | 8.15 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 9.821 | nM | 8.01 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 10.44 | nM | 7.98 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 10.73 | nM | 7.97 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 16.92 | nM | 7.77 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 20.76 | nM | 7.68 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 25.34 | nM | 7.60 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 25.55 | nM | 7.59 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 32.33 | nM | 7.49 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 45.26 | nM | 7.34 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 73.23 | nM | 7.13 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 120.82 | nM | 6.92 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 122.8 | nM | 6.91 |
| CHEMBL217354 | — | IC50 | = | 136.84 | nM | 6.86 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 158.43 | nM | 6.80 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 212.8 | nM | 6.67 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 222.98 | nM | 6.65 |
| CHEMBL803 | CYTARABINE | IC50 | = | 227.86 | nM | 6.64 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 394.25 | nM | 6.40 |
| CHEMBL585951 | — | IC50 | = | 534.53 | nM | 6.27 |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 584.99 | nM | 6.23 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 688.6 | nM | 6.16 |
| CHEMBL1190711 | — | IC50 | = | 980.08 | nM | 6.01 |
| CHEMBL379975 | — | IC50 | = | 1020.55 | nM | 5.99 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1195.76 | nM | 5.92 |
| CHEMBL939 | GEFITINIB | IC50 | = | 1279.18 | nM | 5.89 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1609.23 | nM | 5.79 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 1695.96 | nM | 5.77 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 1822.24 | nM | 5.74 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 2256.53 | nM | 5.65 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 2290.37 | nM | 5.64 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 2722.8 | nM | 5.57 |
| CHEMBL259181 | — | IC50 | = | 3638.3 | nM | 5.44 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 3742.6 | nM | 5.43 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 3827.43 | nM | 5.42 |
| CHEMBL443684 | NAVITOCLAX | IC50 | = | 3895.1 | nM | 5.41 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 4192.37 | nM | 5.38 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 4334.88 | nM | 5.36 |
| CHEMBL591429 | PAC-1 | IC50 | = | 4530.98 | nM | 5.34 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 4888.66 | nM | 5.31 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 4859.26 | nM | 5.31 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 4881.93 | nM | 5.31 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 5867.18 | nM | 5.23 |
| CHEMBL2363137 | — | IC50 | = | 6726.54 | nM | 5.17 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 8250.94 | nM | 5.08 |
| CHEMBL221137 | EMBELIN | IC50 | = | 8470.44 | nM | 5.07 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 12019.02 | nM | 4.92 |