Assay Detail
Functional
CHEMBL2363716
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SANGER: Inhibition of human 8-MG-BA cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | 8-MG-BA |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.75 | 9.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.60 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.23 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.82 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.70 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.47 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.32 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 8.23 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.20 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.10 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.04 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.72 |
| CHEMBL514499 | GW843682X | — | 1 | 7.71 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.66 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.43 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 7.33 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.33 |
| CHEMBL300389 | — | — | 1 | 7.25 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.11 |
| CHEMBL9470 | SHIKONIN | — | 1 | 7.07 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.02 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.98 |
| CHEMBL585951 | — | — | 1 | 6.93 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.91 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.81 |
| CHEMBL217354 | — | — | 1 | 6.81 |
| CHEMBL379300 | A-443654 | — | 1 | 6.79 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.70 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.59 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.2498 | nM | 9.60 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.5889 | nM | 9.23 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.502 | nM | 8.82 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 1.995 | nM | 8.70 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.375 | nM | 8.47 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 4.779 | nM | 8.32 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 5.93 | nM | 8.23 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 6.335 | nM | 8.20 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 7.958 | nM | 8.10 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 9.14 | nM | 8.04 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 18.84 | nM | 7.72 |
| CHEMBL514499 | GW843682X | IC50 | = | 19.37 | nM | 7.71 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 22.12 | nM | 7.66 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 37.25 | nM | 7.43 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 46.87 | nM | 7.33 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 46.29 | nM | 7.33 |
| CHEMBL300389 | — | IC50 | = | 56.0 | nM | 7.25 |
| CHEMBL513909 | BI-2536 | IC50 | = | 58.51 | nM | 7.23 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 78.01 | nM | 7.11 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 85.56 | nM | 7.07 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 94.72 | nM | 7.02 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 104.0 | nM | 6.98 |
| CHEMBL585951 | — | IC50 | = | 116.37 | nM | 6.93 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 123.97 | nM | 6.91 |
| CHEMBL217354 | — | IC50 | = | 153.96 | nM | 6.81 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 154.58 | nM | 6.81 |
| CHEMBL379300 | A-443654 | IC50 | = | 163.01 | nM | 6.79 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 198.1 | nM | 6.70 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 257.68 | nM | 6.59 |
| CHEMBL803 | CYTARABINE | IC50 | = | 340.7 | nM | 6.47 |
| CHEMBL64925 | MG-132 | IC50 | = | 398.37 | nM | 6.40 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 408.43 | nM | 6.39 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 488.95 | nM | 6.31 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 560.56 | nM | 6.25 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 581.52 | nM | 6.24 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1288.66 | nM | 5.89 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 1479.53 | nM | 5.83 |
| CHEMBL379975 | — | IC50 | = | 1553.5 | nM | 5.81 |
| CHEMBL577784 | BX-795 | IC50 | = | 1957.44 | nM | 5.71 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 2019.69 | nM | 5.70 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1982.1 | nM | 5.70 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 2133.74 | nM | 5.67 |
| CHEMBL573107 | — | IC50 | = | 2234.61 | nM | 5.65 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2339.06 | nM | 5.63 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 2532.38 | nM | 5.60 |
| CHEMBL509032 | TAE-684 | IC50 | = | 2654.14 | nM | 5.58 |
| CHEMBL393929 | — | IC50 | = | 3140.49 | nM | 5.50 |
| CHEMBL259181 | — | IC50 | = | 3539.25 | nM | 5.45 |
| CHEMBL221137 | EMBELIN | IC50 | = | 3532.08 | nM | 5.45 |
| CHEMBL191384 | — | IC50 | = | 3677.23 | nM | 5.43 |