Assay Detail
Functional
CHEMBL2363755
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SANGER: Inhibition of human BFTC-905 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BFTC-905 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.78 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 10.30 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 9.85 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 9.57 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 9.18 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.44 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.42 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 8.03 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 7.79 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.69 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 7.33 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.22 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.10 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.03 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 6.96 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 6.89 |
| CHEMBL585951 | — | — | 1 | 6.85 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.60 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 6.59 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.55 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.50 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.39 |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | 6.37 |
| CHEMBL1091644 | LINSITINIB | 3.0 | 1 | 6.33 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.21 |
| CHEMBL217354 | — | — | 1 | 6.15 |
| CHEMBL3349342 | — | — | 1 | 6.14 |
| CHEMBL558642 | GSK-650394 | — | 1 | 6.11 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.11 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.01 |
| CHEMBL577784 | BX-795 | — | 1 | 5.97 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.04994 | nM | 10.30 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 0.1398 | nM | 9.85 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 0.2684 | nM | 9.57 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 0.6625 | nM | 9.18 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.622 | nM | 8.44 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 3.773 | nM | 8.42 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 9.379 | nM | 8.03 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 16.18 | nM | 7.79 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 20.46 | nM | 7.69 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 47.27 | nM | 7.33 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 60.65 | nM | 7.22 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 79.09 | nM | 7.10 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 92.69 | nM | 7.03 |
| CHEMBL803 | CYTARABINE | IC50 | = | 108.31 | nM | 6.96 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 129.16 | nM | 6.89 |
| CHEMBL585951 | — | IC50 | = | 141.2 | nM | 6.85 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 250.02 | nM | 6.60 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 254.58 | nM | 6.59 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 283.61 | nM | 6.55 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 315.21 | nM | 6.50 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 405.26 | nM | 6.39 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 426.21 | nM | 6.37 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 467.58 | nM | 6.33 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 621.26 | nM | 6.21 |
| CHEMBL217354 | — | IC50 | = | 708.18 | nM | 6.15 |
| CHEMBL3349342 | — | IC50 | = | 718.75 | nM | 6.14 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 784.21 | nM | 6.11 |
| CHEMBL558642 | GSK-650394 | IC50 | = | 784.55 | nM | 6.11 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 984.73 | nM | 6.01 |
| CHEMBL577784 | BX-795 | IC50 | = | 1081.01 | nM | 5.97 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 1134.49 | nM | 5.95 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 1242.67 | nM | 5.91 |
| CHEMBL573107 | — | IC50 | = | 1563.32 | nM | 5.81 |
| CHEMBL379975 | — | IC50 | = | 1617.17 | nM | 5.79 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 1880.14 | nM | 5.73 |
| CHEMBL188678 | — | IC50 | = | 2166.87 | nM | 5.66 |
| CHEMBL1190711 | — | IC50 | = | 2294.09 | nM | 5.64 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 2318.88 | nM | 5.63 |
| CHEMBL202721 | — | IC50 | = | 2422.82 | nM | 5.62 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 2423.12 | nM | 5.62 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 2575.48 | nM | 5.59 |
| CHEMBL105442 | CI-1040 | IC50 | = | 2825.3 | nM | 5.55 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 2855.23 | nM | 5.54 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 2901.91 | nM | 5.54 |
| CHEMBL191384 | — | IC50 | = | 3365.07 | nM | 5.47 |
| CHEMBL2363137 | — | IC50 | = | 3645.67 | nM | 5.44 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 4146.49 | nM | 5.38 |
| CHEMBL221137 | EMBELIN | IC50 | = | 5029.55 | nM | 5.30 |
| CHEMBL259181 | — | IC50 | = | 5015.66 | nM | 5.30 |
| CHEMBL472940 | — | IC50 | = | 5147.68 | nM | 5.29 |