Assay Detail
Functional
CHEMBL2363757
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SANGER: Inhibition of human BHT-101 cell growth in a cell viability assay.
99
Total Activities
98
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BHT-101 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 99 | 5.73 | 8.97 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 8.97 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.82 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 8.74 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 8.43 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 8.17 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.01 |
| CHEMBL217354 | — | — | 1 | 7.66 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.52 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.50 |
| CHEMBL803 | CYTARABINE | 4.0 | 1 | 7.38 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.23 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 7.05 |
| CHEMBL3349342 | — | — | 1 | 6.98 |
| CHEMBL1614701 | SELUMETINIB | 4.0 | 1 | 6.97 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 6.71 |
| CHEMBL189963 | PALBOCICLIB | 4.0 | 1 | 6.70 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.68 |
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.61 |
| CHEMBL105442 | CI-1040 | 2.0 | 1 | 6.54 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.50 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.40 |
| CHEMBL1801204 | AZD-8055 | 1.0 | 1 | 6.39 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.33 |
| CHEMBL288441 | BOSUTINIB | 4.0 | 1 | 6.33 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 6.29 |
| CHEMBL1079175 | MK-2206 | 2.0 | 1 | 6.28 |
| CHEMBL521851 | PICTILISIB | 2.0 | 1 | 6.26 |
| CHEMBL255863 | NILOTINIB | 4.0 | 1 | 6.19 |
| CHEMBL585951 | — | — | 1 | 6.18 |
| CHEMBL1230020 | PLX-4720 | — | 1 | 6.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1.063 | nM | 8.97 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 1.519 | nM | 8.82 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 1.822 | nM | 8.74 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 3.72 | nM | 8.43 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 6.704 | nM | 8.17 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 9.799 | nM | 8.01 |
| CHEMBL217354 | — | IC50 | = | 21.83 | nM | 7.66 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 30.05 | nM | 7.52 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 31.36 | nM | 7.50 |
| CHEMBL803 | CYTARABINE | IC50 | = | 41.76 | nM | 7.38 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 58.76 | nM | 7.23 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 88.1 | nM | 7.05 |
| CHEMBL3349342 | — | IC50 | = | 105.62 | nM | 6.98 |
| CHEMBL1614701 | SELUMETINIB | IC50 | = | 106.93 | nM | 6.97 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 197.17 | nM | 6.71 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 198.25 | nM | 6.70 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 210.39 | nM | 6.68 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 244.18 | nM | 6.61 |
| CHEMBL105442 | CI-1040 | IC50 | = | 286.06 | nM | 6.54 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 318.7 | nM | 6.50 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 395.92 | nM | 6.40 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 407.87 | nM | 6.39 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 464.03 | nM | 6.33 |
| CHEMBL288441 | BOSUTINIB | IC50 | = | 465.9 | nM | 6.33 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 513.11 | nM | 6.29 |
| CHEMBL1079175 | MK-2206 | IC50 | = | 529.61 | nM | 6.28 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 544.94 | nM | 6.26 |
| CHEMBL255863 | NILOTINIB | IC50 | = | 642.63 | nM | 6.19 |
| CHEMBL585951 | — | IC50 | = | 666.58 | nM | 6.18 |
| CHEMBL1230020 | PLX-4720 | IC50 | = | 707.02 | nM | 6.15 |
| CHEMBL2134202 | — | IC50 | = | 820.24 | nM | 6.09 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 1147.14 | nM | 5.94 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1159.06 | nM | 5.94 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 1234.9 | nM | 5.91 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1250.23 | nM | 5.90 |
| CHEMBL577784 | BX-795 | IC50 | = | 1578.77 | nM | 5.80 |
| CHEMBL477989 | SB590885 | IC50 | = | 1628.14 | nM | 5.79 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 1740.29 | nM | 5.76 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 2196.54 | nM | 5.66 |
| CHEMBL176544 | — | IC50 | = | 2787.72 | nM | 5.55 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 3107.36 | nM | 5.51 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 3086.07 | nM | 5.51 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 3157.98 | nM | 5.50 |
| CHEMBL188678 | — | IC50 | = | 3599.85 | nM | 5.44 |
| CHEMBL258844 | — | IC50 | = | 4007.04 | nM | 5.40 |
| CHEMBL573107 | — | IC50 | = | 4106.83 | nM | 5.39 |
| CHEMBL11359 | CISPLATIN | IC50 | = | 5822.97 | nM | 5.24 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 6021.5 | nM | 5.22 |
| CHEMBL1173055 | RUCAPARIB | IC50 | = | 6424.73 | nM | 5.19 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 7340.54 | nM | 5.13 |