Assay Detail
Functional
CHEMBL2363767
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SANGER: Inhibition of human Becker cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Becker |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.63 | 8.95 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 8.95 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.74 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.74 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.54 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.27 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.14 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.82 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 7.65 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 7.63 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.52 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 7.47 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.45 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 7.41 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 7.39 |
| CHEMBL300389 | — | — | 1 | 7.32 |
| CHEMBL514499 | GW843682X | — | 1 | 7.22 |
| CHEMBL213100 | — | — | 1 | 7.20 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.19 |
| CHEMBL1201182 | TEMSIROLIMUS | 4.0 | 1 | 7.10 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.87 |
| CHEMBL217354 | — | — | 1 | 6.62 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.57 |
| CHEMBL379300 | A-443654 | — | 1 | 6.52 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.48 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.28 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 6.21 |
| CHEMBL2041933 | AZD-7762 | 1.0 | 1 | 6.18 |
| CHEMBL603469 | LESTAURTINIB | 3.0 | 1 | 6.14 |
| CHEMBL64925 | MG-132 | — | 2 | 6.10 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL159 | VINBLASTINE | IC50 | = | 1.126 | nM | 8.95 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 1.826 | nM | 8.74 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.834 | nM | 8.74 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 2.857 | nM | 8.54 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 5.391 | nM | 8.27 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 7.2 | nM | 8.14 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 15.14 | nM | 7.82 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 22.27 | nM | 7.65 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 23.34 | nM | 7.63 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 30.03 | nM | 7.52 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 34.21 | nM | 7.47 |
| CHEMBL513909 | BI-2536 | IC50 | = | 35.55 | nM | 7.45 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 38.85 | nM | 7.41 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 41.05 | nM | 7.39 |
| CHEMBL300389 | — | IC50 | = | 47.94 | nM | 7.32 |
| CHEMBL514499 | GW843682X | IC50 | = | 59.73 | nM | 7.22 |
| CHEMBL213100 | — | IC50 | = | 63.81 | nM | 7.20 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 64.2 | nM | 7.19 |
| CHEMBL1201182 | TEMSIROLIMUS | IC50 | = | 79.89 | nM | 7.10 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 134.9 | nM | 6.87 |
| CHEMBL217354 | — | IC50 | = | 242.11 | nM | 6.62 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 267.04 | nM | 6.57 |
| CHEMBL379300 | A-443654 | IC50 | = | 303.17 | nM | 6.52 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 334.24 | nM | 6.48 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 521.83 | nM | 6.28 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 616.4 | nM | 6.21 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 658.05 | nM | 6.18 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 723.8 | nM | 6.14 |
| CHEMBL64925 | MG-132 | IC50 | = | 796.21 | nM | 6.10 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 862.32 | nM | 6.06 |
| CHEMBL585951 | — | IC50 | = | 1062.96 | nM | 5.97 |
| CHEMBL803 | CYTARABINE | IC50 | = | 1096.65 | nM | 5.96 |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 1363.15 | nM | 5.87 |
| CHEMBL1801204 | AZD-8055 | IC50 | = | 1521.87 | nM | 5.82 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1582.22 | nM | 5.80 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1642.41 | nM | 5.79 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1803.87 | nM | 5.74 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 1866.63 | nM | 5.73 |
| CHEMBL573107 | — | IC50 | = | 2660.78 | nM | 5.58 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 2694.75 | nM | 5.57 |
| CHEMBL189963 | PALBOCICLIB | IC50 | = | 2958.32 | nM | 5.53 |
| CHEMBL577784 | BX-795 | IC50 | = | 3011.12 | nM | 5.52 |
| CHEMBL64925 | MG-132 | IC50 | = | 3202.54 | nM | 5.50 |
| CHEMBL521851 | PICTILISIB | IC50 | = | 3168.08 | nM | 5.50 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3750.12 | nM | 5.43 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 3928.49 | nM | 5.41 |
| CHEMBL197603 | — | IC50 | = | 4210.27 | nM | 5.38 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 4239.3 | nM | 5.37 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 4373.12 | nM | 5.36 |
| CHEMBL191384 | — | IC50 | = | 4343.86 | nM | 5.36 |