Assay Detail
Functional
CHEMBL2363788
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SANGER: Inhibition of human TE-10 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | TE-10 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.72 | 9.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 9.14 |
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 8.99 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.81 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 8.80 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.60 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 8.48 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 8.44 |
| CHEMBL514499 | GW843682X | — | 1 | 7.90 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 7.79 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.70 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 7.67 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.48 |
| CHEMBL300389 | — | — | 1 | 7.42 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.39 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 7.20 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 7.14 |
| CHEMBL379300 | A-443654 | — | 1 | 7.05 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 7.02 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.95 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.83 |
| CHEMBL585951 | — | — | 1 | 6.51 |
| CHEMBL1972860 | ELESCLOMOL | 3.0 | 1 | 6.50 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.39 |
| CHEMBL109480 | TANESPIMYCIN | 3.0 | 1 | 6.38 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 6.20 |
| CHEMBL509032 | TAE-684 | — | 1 | 6.15 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | — | 1 | 6.14 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 6.11 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.11 |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | 6.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL94657 | PATUPILONE | IC50 | = | 0.7192 | nM | 9.14 |
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 1.03 | nM | 8.99 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 1.543 | nM | 8.81 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 1.573 | nM | 8.80 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 2.536 | nM | 8.60 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 3.296 | nM | 8.48 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 3.625 | nM | 8.44 |
| CHEMBL514499 | GW843682X | IC50 | = | 12.61 | nM | 7.90 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 16.21 | nM | 7.79 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 19.77 | nM | 7.70 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 21.47 | nM | 7.67 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 33.11 | nM | 7.48 |
| CHEMBL300389 | — | IC50 | = | 38.23 | nM | 7.42 |
| CHEMBL513909 | BI-2536 | IC50 | = | 40.46 | nM | 7.39 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 63.57 | nM | 7.20 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 72.6 | nM | 7.14 |
| CHEMBL379300 | A-443654 | IC50 | = | 89.4 | nM | 7.05 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 95.84 | nM | 7.02 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 112.68 | nM | 6.95 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 147.61 | nM | 6.83 |
| CHEMBL585951 | — | IC50 | = | 305.37 | nM | 6.51 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 316.94 | nM | 6.50 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 407.01 | nM | 6.39 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 414.47 | nM | 6.38 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 630.65 | nM | 6.20 |
| CHEMBL509032 | TAE-684 | IC50 | = | 714.96 | nM | 6.15 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 730.32 | nM | 6.14 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 780.39 | nM | 6.11 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 783.12 | nM | 6.11 |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 811.79 | nM | 6.09 |
| CHEMBL2041933 | AZD-7762 | IC50 | = | 909.84 | nM | 6.04 |
| CHEMBL64925 | MG-132 | IC50 | = | 964.3 | nM | 6.02 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 986.09 | nM | 6.01 |
| CHEMBL572878 | TOZASERTIB | IC50 | = | 1129.46 | nM | 5.95 |
| CHEMBL401930 | — | IC50 | = | 1200.47 | nM | 5.92 |
| CHEMBL217354 | — | IC50 | = | 1234.16 | nM | 5.91 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 1281.4 | nM | 5.89 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 1484.35 | nM | 5.83 |
| CHEMBL217092 | SARACATINIB | IC50 | = | 1662.52 | nM | 5.78 |
| CHEMBL1190711 | — | IC50 | = | 1756.04 | nM | 5.75 |
| CHEMBL191384 | — | IC50 | = | 2225.82 | nM | 5.65 |
| CHEMBL535 | SUNITINIB | IC50 | = | 2343.84 | nM | 5.63 |
| CHEMBL197603 | — | IC50 | = | 2356.48 | nM | 5.63 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 2381.02 | nM | 5.62 |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 2708.38 | nM | 5.57 |
| CHEMBL1173655 | AFATINIB | IC50 | = | 2680.78 | nM | 5.57 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 3173.62 | nM | 5.50 |
| CHEMBL554 | LAPATINIB | IC50 | = | 3553.56 | nM | 5.45 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 3920.1 | nM | 5.41 |
| CHEMBL803 | CYTARABINE | IC50 | = | 3908.67 | nM | 5.41 |