Assay Detail
Functional
CHEMBL2363804
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SANGER: Inhibition of human TT cell growth in a cell viability assay.
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | TT |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 38 | 4.97 | 7.94 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 7.94 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.66 |
| CHEMBL9470 | SHIKONIN | — | 1 | 5.77 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 5.64 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 5.59 |
| CHEMBL585951 | — | — | 1 | 5.45 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 5.43 |
| CHEMBL258844 | — | — | 1 | 5.27 |
| CHEMBL477772 | PAZOPANIB | 4.0 | 1 | 5.25 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 5.08 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 5.04 |
| CHEMBL2363137 | — | — | 1 | 5.04 |
| CHEMBL1171837 | PONATINIB | 4.0 | 1 | 4.78 |
| CHEMBL608533 | MIDOSTAURIN | 4.0 | 1 | 4.69 |
| CHEMBL221137 | EMBELIN | — | 1 | 4.63 |
| CHEMBL259181 | — | — | 1 | 4.34 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 4.30 |
| CHEMBL191384 | — | — | 1 | 4.25 |
| CHEMBL512504 | — | — | 1 | 4.25 |
| CHEMBL6067492 | BLEOMYCIN | 4.0 | 1 | 4.23 |
| CHEMBL135561 | — | — | 1 | 4.21 |
| CHEMBL409 | BICALUTAMIDE | 4.0 | 1 | 4.14 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 4.13 |
| CHEMBL1190711 | — | — | 1 | 4.12 |
| CHEMBL575448 | BMS-754807 | 2.0 | 1 | 4.12 |
| CHEMBL1091644 | LINSITINIB | 3.0 | 1 | - |
| CHEMBL44657 | ETOPOSIDE | 4.0 | 1 | - |
| CHEMBL289228 | TIPIFARNIB | 3.0 | 1 | - |
| CHEMBL472004 | — | — | 1 | - |
| CHEMBL412142 | LADUVIGLUSIB | 1.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 11.41 | nM | 7.94 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 216.89 | nM | 6.66 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 1698.76 | nM | 5.77 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 2270.99 | nM | 5.64 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 2580.7 | nM | 5.59 |
| CHEMBL585951 | — | IC50 | = | 3552.04 | nM | 5.45 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 3677.75 | nM | 5.43 |
| CHEMBL258844 | — | IC50 | = | 5327.24 | nM | 5.27 |
| CHEMBL477772 | PAZOPANIB | IC50 | = | 5662.4 | nM | 5.25 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 8330.09 | nM | 5.08 |
| CHEMBL2363137 | — | IC50 | = | 9131.42 | nM | 5.04 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 9069.66 | nM | 5.04 |
| CHEMBL1171837 | PONATINIB | IC50 | = | 16588.77 | nM | 4.78 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 20241.52 | nM | 4.69 |
| CHEMBL221137 | EMBELIN | IC50 | = | 23528.23 | nM | 4.63 |
| CHEMBL259181 | — | IC50 | = | 45140.06 | nM | 4.34 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 49845.94 | nM | 4.30 |
| CHEMBL191384 | — | IC50 | = | 55710.58 | nM | 4.25 |
| CHEMBL512504 | — | IC50 | = | 56771.76 | nM | 4.25 |
| CHEMBL6067492 | BLEOMYCIN | IC50 | = | 59150.08 | nM | 4.23 |
| CHEMBL135561 | — | IC50 | = | 61118.89 | nM | 4.21 |
| CHEMBL409 | BICALUTAMIDE | IC50 | = | 71911.34 | nM | 4.14 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 74634.51 | nM | 4.13 |
| CHEMBL1190711 | — | IC50 | = | 76456.96 | nM | 4.12 |
| CHEMBL575448 | BMS-754807 | IC50 | = | 75325.97 | nM | 4.12 |
| CHEMBL92309 | — | IC50 | = | 537659.79 | nM | - |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 175763.09 | nM | - |
| CHEMBL591429 | PAC-1 | IC50 | = | 230703.42 | nM | - |
| CHEMBL472940 | — | IC50 | = | 2047273.12 | nM | - |
| CHEMBL558642 | GSK-650394 | IC50 | = | 119864.15 | nM | - |
| CHEMBL2165191 | AZD-6482 | IC50 | = | 164985.24 | nM | - |
| CHEMBL1023 | BEXAROTENE | IC50 | = | 679107.88 | nM | - |
| CHEMBL228043 | — | IC50 | = | 546884.7 | nM | - |
| CHEMBL412142 | LADUVIGLUSIB | IC50 | = | 153489.63 | nM | - |
| CHEMBL472004 | — | IC50 | = | 867672.21 | nM | - |
| CHEMBL289228 | TIPIFARNIB | IC50 | = | 123371.48 | nM | - |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 513452.23 | nM | - |
| CHEMBL1091644 | LINSITINIB | IC50 | = | 147250.47 | nM | - |