Assay Detail
Functional
CHEMBL2363830
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SANGER: Inhibition of human no-10 cell growth in a cell viability assay.
139
Total Activities
137
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | no-10 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Genomics of Drug Sensitity in Cancer screening data, Wellcome Trust Sanger Institute
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 139 | 5.41 | 9.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | 3.0 | 1 | 9.68 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 8.44 |
| CHEMBL94657 | PATUPILONE | 3.0 | 1 | 8.26 |
| CHEMBL413 | SIROLIMUS | 4.0 | 1 | 8.14 |
| CHEMBL3545252 | DOCETAXEL | 4.0 | 1 | 8.10 |
| CHEMBL300389 | — | — | 1 | 7.83 |
| CHEMBL1256459 | TORIN1 | — | 1 | 7.80 |
| CHEMBL514499 | GW843682X | — | 1 | 7.68 |
| CHEMBL252164 | LUMINESPIB | 2.0 | 1 | 7.52 |
| CHEMBL553025 | VINORELBINE | 4.0 | 1 | 7.34 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 7.26 |
| CHEMBL64925 | MG-132 | — | 2 | 7.05 |
| CHEMBL379300 | A-443654 | — | 1 | 6.89 |
| CHEMBL53463 | DOXORUBICIN | 4.0 | 1 | 6.79 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.76 |
| CHEMBL888 | GEMCITABINE | 4.0 | 1 | 6.76 |
| CHEMBL1879463 | DACTOLISIB | 3.0 | 1 | 6.70 |
| CHEMBL159 | VINBLASTINE | 4.0 | 1 | 6.57 |
| CHEMBL217354 | — | — | 1 | 6.56 |
| CHEMBL9470 | SHIKONIN | — | 1 | 6.54 |
| CHEMBL105 | MITOMYCIN | 4.0 | 1 | 6.52 |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | 6.50 |
| CHEMBL449158 | BRYOSTATIN 1 | 2.0 | 1 | 6.45 |
| CHEMBL220241 | GSK-269962A | — | 1 | 6.17 |
| CHEMBL96926 | THAPSIGARGIN | — | 1 | 6.11 |
| CHEMBL27759 | ENTINOSTAT | 3.0 | 1 | 5.91 |
| CHEMBL507361 | MIRDAMETINIB | 2.0 | 1 | 5.90 |
| CHEMBL4298697 | — | — | 1 | 5.87 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | 3.0 | 1 | 5.83 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 5.79 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL325041 | BORTEZOMIB | IC50 | = | 0.2098 | nM | 9.68 |
| CHEMBL428647 | PACLITAXEL | IC50 | = | 3.618 | nM | 8.44 |
| CHEMBL94657 | PATUPILONE | IC50 | = | 5.564 | nM | 8.26 |
| CHEMBL413 | SIROLIMUS | IC50 | = | 7.288 | nM | 8.14 |
| CHEMBL3545252 | DOCETAXEL | IC50 | = | 7.881 | nM | 8.10 |
| CHEMBL300389 | — | IC50 | = | 14.78 | nM | 7.83 |
| CHEMBL1256459 | TORIN1 | IC50 | = | 15.84 | nM | 7.80 |
| CHEMBL514499 | GW843682X | IC50 | = | 20.66 | nM | 7.68 |
| CHEMBL252164 | LUMINESPIB | IC50 | = | 30.16 | nM | 7.52 |
| CHEMBL553025 | VINORELBINE | IC50 | = | 45.61 | nM | 7.34 |
| CHEMBL513909 | BI-2536 | IC50 | = | 54.74 | nM | 7.26 |
| CHEMBL64925 | MG-132 | IC50 | = | 89.09 | nM | 7.05 |
| CHEMBL379300 | A-443654 | IC50 | = | 129.02 | nM | 6.89 |
| CHEMBL53463 | DOXORUBICIN | IC50 | = | 160.38 | nM | 6.79 |
| CHEMBL65 | CAMPTOTHECIN | IC50 | = | 174.04 | nM | 6.76 |
| CHEMBL888 | GEMCITABINE | IC50 | = | 173.76 | nM | 6.76 |
| CHEMBL1879463 | DACTOLISIB | IC50 | = | 201.04 | nM | 6.70 |
| CHEMBL159 | VINBLASTINE | IC50 | = | 270.54 | nM | 6.57 |
| CHEMBL217354 | — | IC50 | = | 276.99 | nM | 6.56 |
| CHEMBL9470 | SHIKONIN | IC50 | = | 290.23 | nM | 6.54 |
| CHEMBL105 | MITOMYCIN | IC50 | = | 299.6 | nM | 6.52 |
| CHEMBL5416410 | DASATINIB | IC50 | = | 319.31 | nM | 6.50 |
| CHEMBL449158 | BRYOSTATIN 1 | IC50 | = | 354.99 | nM | 6.45 |
| CHEMBL64925 | MG-132 | IC50 | = | 608.13 | nM | 6.22 |
| CHEMBL220241 | GSK-269962A | IC50 | = | 668.46 | nM | 6.17 |
| CHEMBL96926 | THAPSIGARGIN | IC50 | = | 777.35 | nM | 6.11 |
| CHEMBL27759 | ENTINOSTAT | IC50 | = | 1231.12 | nM | 5.91 |
| CHEMBL507361 | MIRDAMETINIB | IC50 | = | 1264.33 | nM | 5.90 |
| CHEMBL4298697 | — | IC50 | = | 1335.78 | nM | 5.87 |
| CHEMBL2107358 | OBATOCLAX MESYLATE | IC50 | = | 1461.81 | nM | 5.83 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 1617.26 | nM | 5.79 |
| CHEMBL1972860 | ELESCLOMOL | IC50 | = | 1609.82 | nM | 5.79 |
| CHEMBL585951 | — | IC50 | = | 1843.71 | nM | 5.73 |
| CHEMBL392695 | S-TRITYL-L-CYSTEINE | IC50 | = | 1963.65 | nM | 5.71 |
| CHEMBL197603 | — | IC50 | = | 2178.51 | nM | 5.66 |
| CHEMBL109480 | TANESPIMYCIN | IC50 | = | 2549.47 | nM | 5.59 |
| CHEMBL44657 | ETOPOSIDE | IC50 | = | 3488.73 | nM | 5.46 |
| CHEMBL603469 | LESTAURTINIB | IC50 | = | 4994.94 | nM | 5.30 |
| CHEMBL515416 | — | IC50 | = | 6180.21 | nM | 5.21 |
| CHEMBL1084546 | PF-00562271 | IC50 | = | 6478.4 | nM | 5.19 |
| CHEMBL401930 | — | IC50 | = | 6668.57 | nM | 5.18 |
| CHEMBL34259 | METHOTREXATE | IC50 | = | 7307.21 | nM | 5.14 |
| CHEMBL608533 | MIDOSTAURIN | IC50 | = | 9306.33 | nM | 5.03 |
| CHEMBL483847 | — | IC50 | = | 9642.76 | nM | 5.02 |
| CHEMBL1673039 | — | IC50 | = | 9649.23 | nM | 5.02 |
| CHEMBL254129 | CYCLOPAMINE | IC50 | = | 9903.9 | nM | 5.00 |
| CHEMBL1242367 | — | IC50 | = | 10378.0 | nM | 4.98 |
| CHEMBL98 | VORINOSTAT | IC50 | = | 12121.75 | nM | 4.92 |
| CHEMBL2137530 | SERDEMETAN | IC50 | = | 12139.84 | nM | 4.92 |
| CHEMBL213100 | — | IC50 | = | 13143.4 | nM | 4.88 |