Assay Detail
Functional
CHEMBL2379431
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antibacterial activity against Mycobacterium intracellulare ATCC 23068 by alamar blue assay
60
Total Activities
20
Compounds Tested
3
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mycobacterium intracellulare |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Mycobacterium intracellulare (CHEMBL612640) ↗| Type | ORGANISM |
| Organism | Mycobacterium intracellulare |
Publication
Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| MBC | 20 | - | - |
| MIC | 20 | - | - |
| IC50 | 20 | 4.89 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL8 | CIPROFLOXACIN | 4.0 | 3 | 6.00 |
| CHEMBL2376541 | — | — | 3 | 4.40 |
| CHEMBL2376553 | — | — | 3 | 4.28 |
| CHEMBL574091 | — | — | 3 | - |
| CHEMBL2376539 | — | — | 3 | - |
| CHEMBL2376544 | — | — | 3 | - |
| CHEMBL2376552 | — | — | 3 | - |
| CHEMBL2376551 | — | — | 3 | - |
| CHEMBL2376555 | — | — | 3 | - |
| CHEMBL579255 | — | — | 3 | - |
| CHEMBL2376536 | — | — | 3 | - |
| CHEMBL2376557 | — | — | 3 | - |
| CHEMBL2376559 | — | — | 3 | - |
| CHEMBL2376558 | — | — | 3 | - |
| CHEMBL2376690 | — | — | 3 | - |
| CHEMBL2376691 | — | — | 3 | - |
| CHEMBL1373985 | — | — | 3 | - |
| CHEMBL2376692 | — | — | 3 | - |
| CHEMBL1939127 | — | — | 3 | - |
| CHEMBL2376556 | — | — | 3 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL8 | CIPROFLOXACIN | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL2376541 | — | IC50 | = | 39600.0 | nM | 4.40 |
| CHEMBL2376553 | — | IC50 | = | 52900.0 | nM | 4.28 |
| CHEMBL2376541 | — | MIC | = | 41800.0 | nM | - |
| CHEMBL2376536 | — | MIC | - | — | - | |
| CHEMBL8 | CIPROFLOXACIN | MBC | = | 3.02 | uM | - |
| CHEMBL8 | CIPROFLOXACIN | MIC | = | 1510.0 | nM | - |
| CHEMBL2376691 | — | MBC | - | — | - | |
| CHEMBL574091 | — | MBC | - | — | - | |
| CHEMBL2376539 | — | MBC | - | — | - | |
| CHEMBL2376541 | — | MBC | - | — | - | |
| CHEMBL2376544 | — | MBC | - | — | - | |
| CHEMBL2376552 | — | MBC | - | — | - | |
| CHEMBL2376551 | — | MBC | - | — | - | |
| CHEMBL2376553 | — | MBC | - | — | - | |
| CHEMBL2376555 | — | MBC | - | — | - | |
| CHEMBL579255 | — | MBC | - | — | - | |
| CHEMBL2376556 | — | MBC | - | — | - | |
| CHEMBL2376557 | — | MBC | - | — | - | |
| CHEMBL2376559 | — | MBC | - | — | - | |
| CHEMBL2376558 | — | MBC | - | — | - | |
| CHEMBL2376690 | — | MBC | - | — | - | |
| CHEMBL2376536 | — | MBC | - | — | - | |
| CHEMBL1373985 | — | MBC | - | — | - | |
| CHEMBL2376692 | — | MBC | - | — | - | |
| CHEMBL1939127 | — | MBC | - | — | - | |
| CHEMBL2376691 | — | MIC | - | — | - | |
| CHEMBL2376555 | — | IC50 | - | — | - | |
| CHEMBL2376558 | — | MIC | - | — | - | |
| CHEMBL2376551 | — | IC50 | - | — | - | |
| CHEMBL2376552 | — | IC50 | - | — | - | |
| CHEMBL2376544 | — | IC50 | - | — | - | |
| CHEMBL2376539 | — | IC50 | - | — | - | |
| CHEMBL574091 | — | IC50 | - | — | - | |
| CHEMBL2376536 | — | IC50 | - | — | - | |
| CHEMBL1939127 | — | MIC | - | — | - | |
| CHEMBL2376692 | — | MIC | - | — | - | |
| CHEMBL1373985 | — | MIC | - | — | - | |
| CHEMBL1939127 | — | IC50 | - | — | - | |
| CHEMBL2376690 | — | MIC | - | — | - | |
| CHEMBL2376559 | — | MIC | - | — | - | |
| CHEMBL579255 | — | IC50 | - | — | - | |
| CHEMBL2376556 | — | IC50 | - | — | - | |
| CHEMBL2376557 | — | IC50 | - | — | - | |
| CHEMBL2376559 | — | IC50 | - | — | - | |
| CHEMBL2376558 | — | IC50 | - | — | - | |
| CHEMBL2376690 | — | IC50 | - | — | - | |
| CHEMBL2376691 | — | IC50 | - | — | - | |
| CHEMBL1373985 | — | IC50 | - | — | - | |
| CHEMBL2376692 | — | IC50 | - | — | - |