Assay Detail
Binding
CHEMBL2395283
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CGP12177 from human recombinant beta2 adrenergic receptor expressed in CHO cells after 60 mins
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.27 | 9.27 |
| IC50 | 1 | 9.11 | 9.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL452861 | LEVOPROPRANOLOL | 2.0 | 2 | 9.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL452861 | LEVOPROPRANOLOL | Ki | = | 0.54 | nM | 9.27 |
| CHEMBL452861 | LEVOPROPRANOLOL | IC50 | = | 0.78 | nM | 9.11 |