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Assay Detail

CHEMBL2399035

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of DYRK3 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Publication

Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus.
Décor A, Grand-Maître C, Hucke O, O'Meara J, Kuhn C, Constantineau-Forget L, Brochu C, Malenfant E, Bertrand-Laperle M, Bordeleau J, Ghiro E, Pesant M, Fazal G, Gorys V, Little M, Boucher C, Bordeleau S, Turcotte P, Guo T, Garneau M, Spickler C, Gauthier A.
Bioorg Med Chem Lett (2013) 23 : 3841 -3847
PubMed 23726345 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2397315 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2397315 IC50 = 10000.0 nM 5.00