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Assay Detail

CHEMBL2399043

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Functional
Antiviral activity against Poliovirus assessed as protection against virus-induced cytopathic effect by cell-based assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Poliovirus
Confidence 1 — Organism
Curated By Autocuration

Publication

Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus.
Décor A, Grand-Maître C, Hucke O, O'Meara J, Kuhn C, Constantineau-Forget L, Brochu C, Malenfant E, Bertrand-Laperle M, Bordeleau J, Ghiro E, Pesant M, Fazal G, Gorys V, Little M, Boucher C, Bordeleau S, Turcotte P, Guo T, Garneau M, Spickler C, Gauthier A.
Bioorg Med Chem Lett (2013) 23 : 3841 -3847
PubMed 23726345 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 6.33 6.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2397316 1 6.89
CHEMBL2397315 1 6.55
CHEMBL2397314 1 5.96
CHEMBL2397317 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2397316 EC50 = 130.0 nM 6.89
CHEMBL2397315 EC50 = 280.0 nM 6.55
CHEMBL2397314 EC50 = 1100.0 nM 5.96
CHEMBL2397317 EC50 = 1200.0 nM 5.92