Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL2400556

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimigratory activity against human DLD1 cells overexpressing PRL3 by crystal violet staining-based light microscopic analysis
4
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type DLD-1
Confidence 1 — Organism
Curated By Autocuration

Target

DLD-1 (CHEMBL614285)
Type CELL-LINE
Organism Homo sapiens

Publication

Rhodanine-based PRL-3 inhibitors blocked the migration and invasion of metastatic cancer cells.
Min G, Lee SK, Kim HN, Han YM, Lee RH, Jeong DG, Han DC, Kwon BM.
Bioorg Med Chem Lett (2013) 23 : 3769 -3774
PubMed 23726031 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.23 5.30
Inhibition 2 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2397162 2 5.30
CHEMBL207958 2 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2397162 IC50 = 5000.0 nM 5.30
CHEMBL207958 IC50 = 7000.0 nM 5.16
CHEMBL2397162 Inhibition - % -
CHEMBL207958 Inhibition - % -