Assay Detail
Binding
CHEMBL2404444
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Antagonist activity at serotonin 5HT1A receptor (unknown origin) by PDSP assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Selectivity of phenothiazine cholinesterase inhibitors for neurotransmitter systems.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.03 | 6.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL519609 | — | — | 1 | 6.35 |
| CHEMBL240045 | — | — | 1 | 5.96 |
| CHEMBL481153 | — | — | 1 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL519609 | — | Ki | = | 450.0 | nM | 6.35 |
| CHEMBL240045 | — | Ki | = | 1100.0 | nM | 5.96 |
| CHEMBL481153 | — | Ki | = | 1700.0 | nM | 5.77 |