Assay Detail
Binding
CHEMBL2409980
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rabbit muscle glycogen phosphorylase b
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Glycogen phosphorylase, muscle form (CHEMBL4696) ↗| Type | SINGLE PROTEIN |
| Organism | Oryctolagus cuniculus |
Publication
C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 4.68 | 5.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL558445 | — | — | 1 | 5.05 |
| CHEMBL488967 | — | — | 1 | 5.00 |
| CHEMBL600003 | — | — | 1 | 4.80 |
| CHEMBL560324 | — | — | 1 | 4.42 |
| CHEMBL559793 | — | — | 1 | 4.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL558445 | — | Ki | = | 9000.0 | nM | 5.05 |
| CHEMBL488967 | — | Ki | = | 10000.0 | nM | 5.00 |
| CHEMBL600003 | — | Ki | = | 16000.0 | nM | 4.80 |
| CHEMBL560324 | — | Ki | = | 38000.0 | nM | 4.42 |
| CHEMBL559793 | — | Ki | = | 76000.0 | nM | 4.12 |