Assay Detail
Binding
CHEMBL2428811
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human OTR by competitive binding assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Investigation of an F-18 oxytocin receptor selective ligand via PET imaging.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.81 | 7.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2424668 | — | — | 1 | 7.82 |
| CHEMBL2017869 | — | — | 1 | 7.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2424668 | — | Ki | = | 15.0 | nM | 7.82 |
| CHEMBL2017869 | — | Ki | = | 16.0 | nM | 7.80 |