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Assay Detail

CHEMBL2432652

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against KM mouse splenic lymphocytes
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Mus musculus
Cell Type Splenic lymphocyte
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

ADMET (CHEMBL612558)
Type ADMET

Publication

C23 steroids from the venom of Bufo bufo gargarizans.
Tian HY, Luo SL, Liu JS, Wang L, Wang Y, Zhang DM, Zhang XQ, Jiang RW, Ye WC.
J Nat Prod (2013) 76 : 1842 -1847
PubMed 24050254 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 4.10 4.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2431150 1 4.10
CHEMBL250172 BUFOGENIN 2.0 1 -
CHEMBL2431149 1 -
CHEMBL2431148 1 -
CHEMBL2431147 1 -
CHEMBL2429881 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2431150 IC50 = 79400.0 nM 4.10
CHEMBL250172 BUFOGENIN IC50 > 100000.0 nM -
CHEMBL2431149 IC50 > 100000.0 nM -
CHEMBL2431148 IC50 > 100000.0 nM -
CHEMBL2431147 IC50 > 100000.0 nM -
CHEMBL2429881 IC50 > 100000.0 nM -