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Assay Detail

CHEMBL2445842

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Functional
Antioxidant activity assessed as inhibition of H2O2-induced ROS production by DCFH assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 1 — Organism
Curated By Autocuration

Publication

Multifunctional cyclic D,L-α-peptide architectures stimulate non-insulin dependent glucose uptake in skeletal muscle cells and protect them against oxidative stress.
Shapira R, Rudnick S, Daniel B, Viskind O, Aisha V, Richman M, Ayasolla KR, Perelman A, Chill JH, Gruzman A, Rahimipour S.
J Med Chem (2013) 56 : 6709 -6718
PubMed 23984871 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 5 6.26 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3037933 1 6.70
CHEMBL3037934 1 6.52
CHEMBL153 TROLOX 1 6.46
CHEMBL3037932 1 6.40
CHEMBL17962 HISTIDINE 2.0 1 5.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3037933 EC50 = 200.0 nM 6.70
CHEMBL3037934 EC50 = 300.0 nM 6.52
CHEMBL153 TROLOX EC50 = 350.0 nM 6.46
CHEMBL3037932 EC50 = 400.0 nM 6.40
CHEMBL17962 HISTIDINE EC50 = 6000.0 nM 5.22