Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL3047385

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Glycine max (soybean) lipoxygenase using sodium linoleate as substrate
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Glycine max
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Seed linoleate 13S-lipoxygenase-1 (CHEMBL4586)
Type SINGLE PROTEIN
Organism Glycine max

Publication

The novel amidocarbamate derivatives of ketoprofen: synthesis and biological activity.
Rajić Z, Hadjipavlou-Litina D, Pontiki E, Balzarini J, Zorc B.
Med Chem Res (2011) 20 : 210 -219
PubMed 32214761 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.32 4.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1172493 1 4.68
CHEMBL1170394 1 4.50
CHEMBL1172092 1 4.07
CHEMBL1170146 1 4.02
CHEMBL571 KETOPROFEN 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1172493 IC50 = 21000.0 nM 4.68
CHEMBL1170394 IC50 = 32000.0 nM 4.50
CHEMBL1172092 IC50 = 86000.0 nM 4.07
CHEMBL1170146 IC50 = 95000.0 nM 4.02
CHEMBL571 KETOPROFEN IC50 = 130000.0 nM -