Assay Detail
Binding
CHEMBL3056709
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Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleen
21
Total Activities
21
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Spleen |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
In Vitro and In Vivo Characterization of Alpha-1A Selective Agonists and Their Utility for Stress Incontience
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| pEC50 | 11 | - | - |
| EC50 | 10 | 5.53 | 6.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL108804 | — | — | 1 | 6.64 |
| CHEMBL2261346 | — | — | 1 | 6.50 |
| CHEMBL326702 | — | — | 1 | 6.16 |
| CHEMBL323402 | — | — | 1 | 6.01 |
| CHEMBL2261355 | — | — | 1 | 5.42 |
| CHEMBL111554 | — | — | 1 | 5.29 |
| CHEMBL111537 | — | — | 1 | 4.85 |
| CHEMBL109848 | — | — | 1 | 4.84 |
| CHEMBL1076 | DESGLYMIDODRINE | -1.0 | 1 | 4.07 |
| CHEMBL111734 | — | — | 1 | - |
| CHEMBL111536 | — | — | 1 | - |
| CHEMBL320765 | — | — | 1 | - |
| CHEMBL111584 | — | — | 1 | - |
| CHEMBL322492 | — | — | 1 | - |
| CHEMBL111771 | — | — | 1 | - |
| CHEMBL109827 | — | — | 1 | - |
| CHEMBL111391 | — | — | 1 | - |
| CHEMBL321644 | — | — | 1 | - |
| CHEMBL111496 | — | — | 1 | - |
| CHEMBL61006 | PHENYLPROPANOLAMINE | 4.0 | 1 | - |
| CHEMBL325897 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL108804 | — | EC50 | = | 229.09 | nM | 6.64 |
| CHEMBL2261346 | — | EC50 | = | 316.23 | nM | 6.50 |
| CHEMBL326702 | — | EC50 | = | 691.83 | nM | 6.16 |
| CHEMBL323402 | — | EC50 | = | 977.24 | nM | 6.01 |
| CHEMBL2261355 | — | EC50 | = | 3801.89 | nM | 5.42 |
| CHEMBL111554 | — | EC50 | = | 5128.61 | nM | 5.29 |
| CHEMBL111537 | — | EC50 | = | 14125.38 | nM | 4.85 |
| CHEMBL109848 | — | EC50 | = | 14454.4 | nM | 4.84 |
| CHEMBL1076 | DESGLYMIDODRINE | EC50 | = | 85113.8 | nM | 4.07 |
| CHEMBL111734 | — | pEC50 | - | — | - | |
| CHEMBL111536 | — | pEC50 | - | — | - | |
| CHEMBL320765 | — | pEC50 | - | — | - | |
| CHEMBL111584 | — | pEC50 | - | — | - | |
| CHEMBL322492 | — | pEC50 | - | — | - | |
| CHEMBL111771 | — | pEC50 | - | — | - | |
| CHEMBL109827 | — | pEC50 | - | — | - | |
| CHEMBL111391 | — | pEC50 | - | — | - | |
| CHEMBL321644 | — | pEC50 | - | — | - | |
| CHEMBL111496 | — | pEC50 | - | — | - | |
| CHEMBL61006 | PHENYLPROPANOLAMINE | EC50 | = | 281838.29 | nM | - |
| CHEMBL325897 | — | pEC50 | - | — | - |