Assay Detail
Binding
CHEMBL3058307
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to alpha1B adrenoreceptor (unknown origin) by radioligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
(+)-Cyclazosin Derivatives as 1-Adrenoceptor Antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.16 | 9.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2261604 | (+)-CYCLAZOSIN | — | 1 | 9.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2261604 | (+)-CYCLAZOSIN | Ki | = | 0.6918 | nM | 9.16 |