Assay Detail
Binding
CHEMBL3068024
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Uncompetitive inhibition of yeast alpha-glucosidase by Lineweaver-Burk plot analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Saccharomyces cerevisiae |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and structureactivity relationships of serotonin derivatives effect on -glucosidase inhibition
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.14 | 4.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL559089 | N-CAFFEOYLSEROTONIN | — | 1 | 4.19 |
| CHEMBL1760547 | N-P-COUMAROYL SEROTONIN | — | 1 | 4.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL559089 | N-CAFFEOYLSEROTONIN | Ki | = | 64400.0 | nM | 4.19 |
| CHEMBL1760547 | N-P-COUMAROYL SEROTONIN | Ki | = | 81600.0 | nM | 4.09 |