Assay Detail
Binding
CHEMBL3082041
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]EBOB from GABA receptor in Musca domestica (house fly) head P2 membrane after 70 min by liquid scintillation counting
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Musca domestica |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Isocoumarin Derivative as a Novel GABA Receptor Ligand from Neosartorya quadricincta
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.06 | 7.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1684587 | — | — | 1 | 7.06 |
| CHEMBL2269235 | DIHYDROISOCOUMARIN | — | 1 | 7.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1684587 | — | IC50 | = | 88.0 | nM | 7.06 |
| CHEMBL2269235 | DIHYDROISOCOUMARIN | IC50 | = | 88.0 | nM | 7.06 |