Assay Detail
Binding
CHEMBL3089444
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Agonist activity at S1P4 receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Modulators of the Sphingosine 1-phosphate receptor 1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.07 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL314854 | FINGOLIMOD | 4.0 | 1 | 9.52 |
| CHEMBL3086703 | — | — | 1 | 6.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL314854 | FINGOLIMOD | EC50 | = | 0.3 | nM | 9.52 |
| CHEMBL3086703 | — | EC50 | = | 245.0 | nM | 6.61 |