Assay Detail
Binding
CHEMBL3096274
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Inhibition of full-length Mps1 kinase (unknown origin)
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel Mps1 kinase inhibitors: from purine to pyrrolopyrimidine and quinazoline leads.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 7.94 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2047959 | — | — | 1 | 8.70 |
| CHEMBL3092039 | — | — | 1 | 8.70 |
| CHEMBL3092037 | — | — | 1 | 8.30 |
| CHEMBL2047943 | — | — | 1 | 8.30 |
| CHEMBL3092038 | — | — | 1 | 8.10 |
| CHEMBL3092036 | — | — | 1 | 8.05 |
| CHEMBL3092035 | — | — | 1 | 7.92 |
| CHEMBL3092030 | — | — | 1 | 7.70 |
| CHEMBL3092029 | — | — | 1 | 7.66 |
| CHEMBL3092026 | — | — | 1 | 7.55 |
| CHEMBL3092032 | — | — | 1 | 7.50 |
| CHEMBL3092025 | — | — | 1 | 7.46 |
| CHEMBL3092028 | — | — | 1 | 7.34 |
| CHEMBL3092034 | — | — | 1 | - |
| CHEMBL3091469 | — | — | 1 | - |
| CHEMBL3092033 | — | — | 1 | - |
| CHEMBL3092031 | — | — | 1 | - |
| CHEMBL3092027 | — | — | 1 | - |
| CHEMBL3092024 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2047959 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3092039 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3092037 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL2047943 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL3092038 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL3092036 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL3092035 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL3092030 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3092029 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL3092026 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL3092032 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL3092025 | — | IC50 | = | 35.0 | nM | 7.46 |
| CHEMBL3092028 | — | IC50 | = | 46.0 | nM | 7.34 |
| CHEMBL3092034 | — | IC50 | > | 100.0 | nM | - |
| CHEMBL3091469 | — | IC50 | > | 100.0 | nM | - |
| CHEMBL3092033 | — | IC50 | > | 100.0 | nM | - |
| CHEMBL3092031 | — | IC50 | > | 100.0 | nM | - |
| CHEMBL3092027 | — | IC50 | > | 100.0 | nM | - |
| CHEMBL3092024 | — | IC50 | > | 100.0 | nM | - |