Assay Detail
Binding
CHEMBL3096539
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of pig/bovine heart myocardium PDE2 after 15 mins by scintillation proximity assay in presence of [3H]-cAMP
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Myocardium |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PDE2 inhibition: potential for the treatment of cognitive disorders.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.70 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL370962 | — | — | 1 | 8.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL370962 | — | IC50 | = | 2.0 | nM | 8.70 |