Assay Detail
Functional
CHEMBL3101585
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Antiproliferative activity against human HL60 cells
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
NAD-based inhibitors with anticancer potential.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 4.79 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3098181 | — | — | 1 | 5.68 |
| CHEMBL3098174 | — | — | 1 | 5.35 |
| CHEMBL3098170 | — | — | 1 | 5.33 |
| CHEMBL3098164 | — | — | 1 | 5.08 |
| CHEMBL3098180 | — | — | 1 | 5.03 |
| CHEMBL3098172 | — | — | 1 | 4.75 |
| CHEMBL2437258 | — | — | 1 | 4.66 |
| CHEMBL2437261 | — | — | 1 | 4.51 |
| CHEMBL3098167 | — | — | 1 | 4.46 |
| CHEMBL2437265 | — | — | 1 | 4.46 |
| CHEMBL2437262 | — | — | 1 | 4.44 |
| CHEMBL2437266 | — | — | 1 | 4.39 |
| CHEMBL2437272 | — | — | 1 | 4.14 |
| CHEMBL3098169 | — | — | 1 | - |
| CHEMBL3098168 | — | — | 1 | - |
| CHEMBL3098166 | — | — | 1 | - |
| CHEMBL3098165 | — | — | 1 | - |
| CHEMBL3098163 | — | — | 1 | - |
| CHEMBL2437255 | — | — | 1 | - |
| CHEMBL3098186 | — | — | 1 | - |
| CHEMBL2437254 | — | — | 1 | - |
| CHEMBL3098185 | — | — | 1 | - |
| CHEMBL2437269 | — | — | 1 | - |
| CHEMBL3098184 | — | — | 1 | - |
| CHEMBL2437273 | — | — | 1 | - |
| CHEMBL3098183 | — | — | 1 | - |
| CHEMBL3098182 | — | — | 1 | - |
| CHEMBL3098173 | — | — | 1 | - |
| CHEMBL3098171 | — | — | 1 | - |
| CHEMBL3098175 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3098181 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL3098174 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL3098170 | — | IC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL3098164 | — | IC50 | = | 8300.0 | nM | 5.08 |
| CHEMBL3098180 | — | IC50 | = | 9300.0 | nM | 5.03 |
| CHEMBL3098172 | — | IC50 | = | 18000.0 | nM | 4.75 |
| CHEMBL2437258 | — | IC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL2437261 | — | IC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL3098167 | — | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL2437265 | — | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL2437262 | — | IC50 | = | 36000.0 | nM | 4.44 |
| CHEMBL2437266 | — | IC50 | = | 41000.0 | nM | 4.39 |
| CHEMBL2437272 | — | IC50 | = | 72000.0 | nM | 4.14 |
| CHEMBL3098169 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098168 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098166 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098165 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098163 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437255 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098186 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437254 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098185 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437269 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098184 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2437273 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098183 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098182 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098173 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098171 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3098175 | — | IC50 | > | 100000.0 | nM | - |