Assay Detail
Functional
CHEMBL3107427
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human RCC4 cells after 4 days by XTT assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | RCC4 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identifying novel targets in renal cell carcinoma: design and synthesis of affinity chromatography reagents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 5.69 | 6.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3105156 | — | — | 1 | 6.80 |
| CHEMBL3105157 | — | — | 1 | 5.77 |
| CHEMBL565269 | — | — | 1 | 5.68 |
| CHEMBL3105160 | — | — | 1 | 5.54 |
| CHEMBL3105162 | — | — | 1 | 5.24 |
| CHEMBL3105163 | — | — | 1 | 5.10 |
| CHEMBL3105164 | — | — | 1 | - |
| CHEMBL3105161 | — | — | 1 | - |
| CHEMBL3105159 | — | — | 1 | - |
| CHEMBL3105158 | — | — | 1 | - |
| CHEMBL3105170 | — | — | 1 | - |
| CHEMBL3105169 | — | — | 1 | - |
| CHEMBL3105168 | — | — | 1 | - |
| CHEMBL3105167 | — | — | 1 | - |
| CHEMBL3105166 | — | — | 1 | - |
| CHEMBL3105165 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3105156 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL3105157 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL565269 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL3105160 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL3105162 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL3105163 | — | IC50 | = | 7900.0 | nM | 5.10 |
| CHEMBL3105164 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3105161 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3105159 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3105158 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3105170 | — | IC50 | < | 1000.0 | nM | - |
| CHEMBL3105169 | — | IC50 | < | 1000.0 | nM | - |
| CHEMBL3105168 | — | IC50 | < | 1000.0 | nM | - |
| CHEMBL3105167 | — | IC50 | < | 1000.0 | nM | - |
| CHEMBL3105166 | — | IC50 | < | 1000.0 | nM | - |
| CHEMBL3105165 | — | IC50 | < | 1000.0 | nM | - |