Assay Detail
Functional
CHEMBL3110669
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Cytotoxicity against human 67EF cells assessed as cell viability after 3 days by Alamar Blue assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Potent Targeting of the STAT3 Protein in Brain Cancer Stem Cells: A Promising Route for Treating Glioblastoma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.67 | 6.97 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3108909 | — | — | 1 | 6.97 |
| CHEMBL3108911 | — | — | 1 | 6.67 |
| CHEMBL3108910 | — | — | 1 | 6.67 |
| CHEMBL3108782 | — | — | 1 | 6.36 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3108909 | — | IC50 | = | 106.0 | nM | 6.97 |
| CHEMBL3108911 | — | IC50 | = | 214.0 | nM | 6.67 |
| CHEMBL3108910 | — | IC50 | = | 214.5 | nM | 6.67 |
| CHEMBL3108782 | — | IC50 | = | 435.5 | nM | 6.36 |