Assay Detail
Functional
CHEMBL3112094
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Cytotoxicity against human JeKo1 cells after 72 hrs by CellTiter-Glo assay
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | JeKo-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Optimization of antitumor modulators of pre-mRNA splicing.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 6.37 | 7.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3108948 | — | — | 1 | 7.66 |
| CHEMBL3108947 | — | — | 1 | 7.39 |
| CHEMBL3108950 | — | — | 1 | 7.00 |
| CHEMBL566107 | — | — | 1 | 6.66 |
| CHEMBL3108944 | — | — | 1 | 6.52 |
| CHEMBL3108951 | — | — | 1 | 6.47 |
| CHEMBL3108935 | — | — | 1 | 6.21 |
| CHEMBL3108937 | — | — | 1 | 6.16 |
| CHEMBL3108938 | — | — | 1 | 6.16 |
| CHEMBL3108939 | — | — | 1 | 6.11 |
| CHEMBL3108945 | — | — | 1 | 6.05 |
| CHEMBL3108943 | — | — | 1 | 6.03 |
| CHEMBL3108942 | — | — | 1 | 6.01 |
| CHEMBL3108940 | — | — | 1 | 5.88 |
| CHEMBL3108941 | — | — | 1 | 5.83 |
| CHEMBL3108946 | — | — | 1 | 5.72 |
| CHEMBL3108936 | — | — | 1 | - |
| CHEMBL3108932 | — | — | 1 | - |
| CHEMBL3108933 | — | — | 1 | - |
| CHEMBL3108934 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3108948 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL3108947 | — | IC50 | = | 41.0 | nM | 7.39 |
| CHEMBL3108950 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL566107 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL3108944 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL3108951 | — | IC50 | = | 340.0 | nM | 6.47 |
| CHEMBL3108935 | — | IC50 | = | 610.0 | nM | 6.21 |
| CHEMBL3108937 | — | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL3108938 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL3108939 | — | IC50 | = | 780.0 | nM | 6.11 |
| CHEMBL3108945 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL3108943 | — | IC50 | = | 940.0 | nM | 6.03 |
| CHEMBL3108942 | — | IC50 | = | 970.0 | nM | 6.01 |
| CHEMBL3108940 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL3108941 | — | IC50 | = | 1470.0 | nM | 5.83 |
| CHEMBL3108946 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL3108936 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL3108932 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL3108933 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL3108934 | — | IC50 | > | 1000.0 | nM | - |