Assay Detail
Functional
CHEMBL3135045
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Antiprotozoal activity against Plasmodium falciparum D6 assessed as growth inhibition after 72 hrs by SYBR Green dye-based fluorescence assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Plasmodium falciparum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 6.68 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL514409 | HESPERADIN | — | 1 | 8.00 |
| CHEMBL3134085 | — | — | 1 | 7.28 |
| CHEMBL3134095 | — | — | 1 | 7.27 |
| CHEMBL3134087 | — | — | 1 | 7.17 |
| CHEMBL3134086 | — | — | 1 | 6.97 |
| CHEMBL3134093 | — | — | 1 | 6.96 |
| CHEMBL3134091 | — | — | 1 | 6.78 |
| CHEMBL3134005 | — | — | 1 | 6.70 |
| CHEMBL3134004 | — | — | 1 | 6.66 |
| CHEMBL500435 | — | — | 1 | 6.64 |
| CHEMBL3134090 | — | — | 1 | 6.63 |
| CHEMBL3134088 | — | — | 1 | 6.62 |
| CHEMBL3134003 | — | — | 1 | 6.56 |
| CHEMBL3134096 | — | — | 1 | 6.22 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | 6.08 |
| CHEMBL402548 | DANUSERTIB | 2.0 | 1 | 6.07 |
| CHEMBL3134089 | — | — | 1 | 5.87 |
| CHEMBL3134094 | — | — | 1 | 5.79 |
| CHEMBL3134092 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL514409 | HESPERADIN | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL3134085 | — | EC50 | = | 52.0 | nM | 7.28 |
| CHEMBL3134095 | — | EC50 | = | 54.0 | nM | 7.27 |
| CHEMBL3134087 | — | EC50 | = | 68.0 | nM | 7.17 |
| CHEMBL3134086 | — | EC50 | = | 107.0 | nM | 6.97 |
| CHEMBL3134093 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL3134091 | — | EC50 | = | 167.0 | nM | 6.78 |
| CHEMBL3134005 | — | EC50 | = | 199.0 | nM | 6.70 |
| CHEMBL3134004 | — | EC50 | = | 218.0 | nM | 6.66 |
| CHEMBL500435 | — | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL3134090 | — | EC50 | = | 233.0 | nM | 6.63 |
| CHEMBL3134088 | — | EC50 | = | 241.0 | nM | 6.62 |
| CHEMBL3134003 | — | EC50 | = | 275.0 | nM | 6.56 |
| CHEMBL3134096 | — | EC50 | = | 595.0 | nM | 6.22 |
| CHEMBL572878 | TOZASERTIB | EC50 | = | 838.0 | nM | 6.08 |
| CHEMBL402548 | DANUSERTIB | EC50 | = | 857.0 | nM | 6.07 |
| CHEMBL3134089 | — | EC50 | = | 1364.0 | nM | 5.87 |
| CHEMBL3134094 | — | EC50 | = | 1607.0 | nM | 5.79 |
| CHEMBL3134092 | — | EC50 | > | 15000.0 | nM | - |