Assay Detail
Functional
CHEMBL3135046
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Antiprotozoal activity against intracellular amastigote stage of Leishmania major infected in mouse RAW246.7 cells assessed as growth inhibition after 96 hrs by luciferase reporter gene assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Leishmania major |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 5.70 | 5.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3134095 | — | — | 1 | 5.78 |
| CHEMBL3134086 | — | — | 1 | 5.72 |
| CHEMBL3134003 | — | — | 1 | 5.69 |
| CHEMBL514409 | HESPERADIN | — | 1 | 5.62 |
| CHEMBL572878 | TOZASERTIB | 2.0 | 1 | - |
| CHEMBL3134094 | — | — | 1 | - |
| CHEMBL3134093 | — | — | 1 | - |
| CHEMBL3134092 | — | — | 1 | - |
| CHEMBL3134091 | — | — | 1 | - |
| CHEMBL3134090 | — | — | 1 | - |
| CHEMBL3134089 | — | — | 1 | - |
| CHEMBL402548 | DANUSERTIB | 2.0 | 1 | - |
| CHEMBL3134085 | — | — | 1 | - |
| CHEMBL3134005 | — | — | 1 | - |
| CHEMBL500435 | — | — | 1 | - |
| CHEMBL3134004 | — | — | 1 | - |
| CHEMBL3134087 | — | — | 1 | - |
| CHEMBL3134096 | — | — | 1 | - |
| CHEMBL3134088 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3134095 | — | EC50 | = | 1680.0 | nM | 5.78 |
| CHEMBL3134086 | — | EC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL3134003 | — | EC50 | = | 2040.0 | nM | 5.69 |
| CHEMBL514409 | HESPERADIN | EC50 | = | 2370.0 | nM | 5.62 |
| CHEMBL572878 | TOZASERTIB | EC50 | - | — | - | |
| CHEMBL3134094 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134093 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134092 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134091 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134090 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134089 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL402548 | DANUSERTIB | EC50 | - | — | - | |
| CHEMBL3134085 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134005 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL500435 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134004 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134087 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134096 | — | EC50 | > | 4000.0 | nM | - |
| CHEMBL3134088 | — | EC50 | > | 4000.0 | nM | - |