Assay Detail
Binding
CHEMBL3214794
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Counterscreen for inhibitors of Crimean-Congo Hemorrhagic Fever (CCHF) viral ovarian tumor domain protease (vOTU): Pep-AMC substrate: Fluorescence-based biochemical high throughput screening assay to identify inhibitors of Crimean-Congo Hemorrhagic Fever (CCHF) viral ovarian tumor domain protease (vOTU): Ub-AMC substrate. (Class of assay: confirmatory)
226
Total Activities
226
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 226 | 4.97 | 6.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1734083 | — | — | 1 | 6.41 |
| CHEMBL599924 | — | — | 1 | 6.31 |
| CHEMBL1999630 | — | — | 1 | 6.27 |
| CHEMBL1210769 | — | — | 1 | 6.22 |
| CHEMBL1384253 | — | — | 1 | 6.18 |
| CHEMBL1728280 | — | — | 1 | 6.07 |
| CHEMBL1998302 | — | — | 1 | 5.99 |
| CHEMBL3189714 | — | — | 1 | 5.98 |
| CHEMBL1163377 | — | — | 1 | 5.97 |
| CHEMBL1359236 | — | — | 1 | 5.97 |
| CHEMBL1735482 | — | — | 1 | 5.96 |
| CHEMBL1598762 | — | — | 1 | 5.95 |
| CHEMBL1463659 | — | — | 1 | 5.94 |
| CHEMBL2003651 | — | — | 1 | 5.91 |
| CHEMBL1466516 | — | — | 1 | 5.88 |
| CHEMBL3191855 | — | — | 1 | 5.88 |
| CHEMBL1505544 | — | — | 1 | 5.88 |
| CHEMBL1719244 | — | — | 1 | 5.87 |
| CHEMBL1877709 | — | — | 1 | 5.85 |
| CHEMBL1453503 | — | — | 1 | 5.84 |
| CHEMBL1733422 | — | — | 1 | 5.83 |
| CHEMBL1331912 | — | — | 1 | 5.82 |
| CHEMBL3196451 | — | — | 1 | 5.75 |
| CHEMBL3191689 | — | — | 1 | 5.74 |
| CHEMBL1982305 | — | — | 1 | 5.70 |
| CHEMBL1335844 | — | — | 1 | 5.67 |
| CHEMBL339561 | — | — | 1 | 5.65 |
| CHEMBL1969046 | — | — | 1 | 5.63 |
| CHEMBL1546172 | — | — | 1 | 5.62 |
| CHEMBL3190880 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1734083 | — | IC50 | = | 387.44 | nM | 6.41 |
| CHEMBL599924 | — | IC50 | = | 487.0 | nM | 6.31 |
| CHEMBL1999630 | — | IC50 | = | 535.73 | nM | 6.27 |
| CHEMBL1210769 | — | IC50 | = | 596.74 | nM | 6.22 |
| CHEMBL1384253 | — | IC50 | = | 662.32 | nM | 6.18 |
| CHEMBL1728280 | — | IC50 | = | 853.3 | nM | 6.07 |
| CHEMBL1998302 | — | IC50 | = | 1031.0 | nM | 5.99 |
| CHEMBL3189714 | — | IC50 | = | 1043.0 | nM | 5.98 |
| CHEMBL1359236 | — | IC50 | = | 1066.0 | nM | 5.97 |
| CHEMBL1163377 | — | IC50 | = | 1075.0 | nM | 5.97 |
| CHEMBL1735482 | — | IC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL1598762 | — | IC50 | = | 1131.0 | nM | 5.95 |
| CHEMBL1463659 | — | IC50 | = | 1157.0 | nM | 5.94 |
| CHEMBL2003651 | — | IC50 | = | 1239.0 | nM | 5.91 |
| CHEMBL1505544 | — | IC50 | = | 1334.0 | nM | 5.88 |
| CHEMBL1466516 | — | IC50 | = | 1305.0 | nM | 5.88 |
| CHEMBL3191855 | — | IC50 | = | 1335.0 | nM | 5.88 |
| CHEMBL1719244 | — | IC50 | = | 1365.0 | nM | 5.87 |
| CHEMBL1877709 | — | IC50 | = | 1401.0 | nM | 5.85 |
| CHEMBL1453503 | — | IC50 | = | 1446.0 | nM | 5.84 |
| CHEMBL1733422 | — | IC50 | = | 1493.0 | nM | 5.83 |
| CHEMBL1331912 | — | IC50 | = | 1505.0 | nM | 5.82 |
| CHEMBL3196451 | — | IC50 | = | 1792.0 | nM | 5.75 |
| CHEMBL3191689 | — | IC50 | = | 1813.0 | nM | 5.74 |
| CHEMBL1982305 | — | IC50 | = | 1991.0 | nM | 5.70 |
| CHEMBL1335844 | — | IC50 | = | 2157.0 | nM | 5.67 |
| CHEMBL339561 | — | IC50 | = | 2231.0 | nM | 5.65 |
| CHEMBL1969046 | — | IC50 | = | 2359.0 | nM | 5.63 |
| CHEMBL1546172 | — | IC50 | = | 2369.0 | nM | 5.62 |
| CHEMBL3190880 | — | IC50 | = | 2509.0 | nM | 5.60 |
| CHEMBL57013 | — | IC50 | = | 2578.0 | nM | 5.59 |
| CHEMBL284328 | HOMIDIUM BROMIDE | IC50 | = | 3321.0 | nM | 5.48 |
| CHEMBL1716155 | — | IC50 | = | 3646.0 | nM | 5.44 |
| CHEMBL51931 | 9,10-PHENANTHRENEQUINONE | IC50 | = | 3748.0 | nM | 5.43 |
| CHEMBL1471498 | — | IC50 | = | 4040.0 | nM | 5.39 |
| CHEMBL1724452 | — | IC50 | = | 4138.0 | nM | 5.38 |
| CHEMBL1438881 | — | IC50 | = | 4196.0 | nM | 5.38 |
| CHEMBL1709564 | — | IC50 | = | 4332.0 | nM | 5.36 |
| CHEMBL1698802 | — | IC50 | = | 4325.0 | nM | 5.36 |
| CHEMBL3197091 | — | IC50 | = | 4540.0 | nM | 5.34 |
| CHEMBL3216654 | — | IC50 | = | 4596.0 | nM | 5.34 |
| CHEMBL1723968 | — | IC50 | = | 4574.0 | nM | 5.34 |
| CHEMBL1964407 | — | IC50 | = | 4609.0 | nM | 5.34 |
| CHEMBL1302524 | — | IC50 | = | 4768.0 | nM | 5.32 |
| CHEMBL156174 | — | IC50 | = | 4940.0 | nM | 5.31 |
| CHEMBL1702473 | — | IC50 | = | 4983.0 | nM | 5.30 |
| CHEMBL1555938 | — | IC50 | = | 5106.0 | nM | 5.29 |
| CHEMBL1706454 | — | IC50 | = | 5160.0 | nM | 5.29 |
| CHEMBL1589737 | — | IC50 | = | 5201.0 | nM | 5.28 |
| CHEMBL2141749 | — | IC50 | = | 5367.0 | nM | 5.27 |