Assay Detail
Functional
CHEMBL3214907
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PubChem BioAssay. Dose Response confirmation of small molecule inhibitors originally identified via uHTS of Artemis endonuclease activity via a fluorescence intensity assay. (Class of assay: confirmatory)
133
Total Activities
133
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 133 | 5.17 | 6.01 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1583339 | — | — | 1 | 6.01 |
| CHEMBL1421559 | — | — | 1 | 5.95 |
| CHEMBL1340032 | — | — | 1 | 5.91 |
| CHEMBL1525442 | — | — | 1 | 5.85 |
| CHEMBL1470135 | — | — | 1 | 5.83 |
| CHEMBL3197433 | — | — | 1 | 5.82 |
| CHEMBL1526649 | — | — | 1 | 5.80 |
| CHEMBL1410497 | — | — | 1 | 5.78 |
| CHEMBL1979849 | — | — | 1 | 5.72 |
| CHEMBL1503307 | — | — | 1 | 5.71 |
| CHEMBL1575622 | — | — | 1 | 5.68 |
| CHEMBL1542862 | — | — | 1 | 5.66 |
| CHEMBL3192616 | — | — | 1 | 5.65 |
| CHEMBL3192592 | — | — | 1 | 5.58 |
| CHEMBL1550490 | — | — | 1 | 5.58 |
| CHEMBL1461574 | — | — | 1 | 5.50 |
| CHEMBL1391287 | — | — | 1 | 5.45 |
| CHEMBL3190629 | — | — | 1 | 5.44 |
| CHEMBL3199553 | — | — | 1 | 5.44 |
| CHEMBL1533366 | — | — | 1 | 5.42 |
| CHEMBL1464065 | — | — | 1 | 5.34 |
| CHEMBL1443205 | — | — | 1 | 5.33 |
| CHEMBL1378339 | — | — | 1 | 5.33 |
| CHEMBL3193098 | — | — | 1 | 5.33 |
| CHEMBL1448732 | — | — | 1 | 5.30 |
| CHEMBL1330556 | — | — | 1 | 5.23 |
| CHEMBL1372855 | — | — | 1 | 5.22 |
| CHEMBL3196345 | — | — | 1 | 5.19 |
| CHEMBL3197459 | — | — | 1 | 5.18 |
| CHEMBL1386272 | — | — | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1583339 | — | IC50 | = | 967.0 | nM | 6.01 |
| CHEMBL1421559 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1340032 | — | IC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL1525442 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL1470135 | — | IC50 | = | 1480.0 | nM | 5.83 |
| CHEMBL3197433 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL1526649 | — | IC50 | = | 1590.0 | nM | 5.80 |
| CHEMBL1410497 | — | IC50 | = | 1680.0 | nM | 5.78 |
| CHEMBL1979849 | — | IC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL1503307 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL1575622 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1542862 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL3192616 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1550490 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL3192592 | — | IC50 | = | 2650.0 | nM | 5.58 |
| CHEMBL1461574 | — | IC50 | = | 3190.0 | nM | 5.50 |
| CHEMBL1391287 | — | IC50 | = | 3590.0 | nM | 5.45 |
| CHEMBL3190629 | — | IC50 | = | 3640.0 | nM | 5.44 |
| CHEMBL3199553 | — | IC50 | = | 3620.0 | nM | 5.44 |
| CHEMBL1533366 | — | IC50 | = | 3810.0 | nM | 5.42 |
| CHEMBL1464065 | — | IC50 | = | 4520.0 | nM | 5.34 |
| CHEMBL1443205 | — | IC50 | = | 4710.0 | nM | 5.33 |
| CHEMBL3193098 | — | IC50 | = | 4680.0 | nM | 5.33 |
| CHEMBL1378339 | — | IC50 | = | 4650.0 | nM | 5.33 |
| CHEMBL1448732 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL1330556 | — | IC50 | = | 5840.0 | nM | 5.23 |
| CHEMBL1372855 | — | IC50 | = | 6030.0 | nM | 5.22 |
| CHEMBL3196345 | — | IC50 | = | 6460.0 | nM | 5.19 |
| CHEMBL3197459 | — | IC50 | = | 6570.0 | nM | 5.18 |
| CHEMBL1386272 | — | IC50 | = | 6960.0 | nM | 5.16 |
| CHEMBL2000196 | — | IC50 | = | 7400.0 | nM | 5.13 |
| CHEMBL1579841 | — | IC50 | = | 7470.0 | nM | 5.13 |
| CHEMBL1324113 | — | IC50 | = | 7660.0 | nM | 5.12 |
| CHEMBL1445776 | — | IC50 | = | 7750.0 | nM | 5.11 |
| CHEMBL1466712 | — | IC50 | = | 8960.0 | nM | 5.05 |
| CHEMBL1587783 | — | IC50 | = | 9250.0 | nM | 5.03 |
| CHEMBL1377648 | — | IC50 | = | 9580.0 | nM | 5.02 |
| CHEMBL1559375 | — | IC50 | = | 9490.0 | nM | 5.02 |
| CHEMBL1563484 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL1967586 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL1390659 | — | IC50 | = | 11500.0 | nM | 4.94 |
| CHEMBL1330307 | — | IC50 | = | 11400.0 | nM | 4.94 |
| CHEMBL1699206 | — | IC50 | = | 11400.0 | nM | 4.94 |
| CHEMBL1496007 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL1532645 | — | IC50 | = | 11800.0 | nM | 4.93 |
| CHEMBL1560141 | — | IC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL1404929 | — | IC50 | = | 13300.0 | nM | 4.88 |
| CHEMBL1449173 | — | IC50 | = | 14400.0 | nM | 4.84 |
| CHEMBL1519843 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL3192181 | — | IC50 | = | 15500.0 | nM | 4.81 |