Assay Detail
Binding
CHEMBL3223401
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Inhibition of c-FOS/AP1 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Small-molecule inhibitors of dimeric transcription factors: Antagonism of proteinprotein and proteinDNA interactions
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.10 | 5.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3222140 | — | — | 1 | 5.10 |
| CHEMBL3222137 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3222140 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL3222137 | — | IC50 | = | 200000.0 | nM | - |