Assay Detail
Binding
CHEMBL3226052
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of methicillin-resistant Staphylococcus aureus DHFR F98Y/H30N double mutant
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Staphylococcus aureus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Antifolates as effective antimicrobial agents: new generations of trimethoprim analogs
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.96 | 6.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL520358 | — | — | 1 | 6.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL520358 | — | Ki | = | 110.0 | nM | 6.96 |