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Assay Detail

CHEMBL3243189

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HL60 cells after 24 hrs by WST-1 assay
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HL-60
Confidence 1 — Organism
Curated By Autocuration

Target

HL-60 (CHEMBL383)
Type CELL-LINE
Organism Homo sapiens

Publication

Cytotoxic constituents from Lobaria scrobiculata and a comparison of two bioassays for their evaluation.
Schinkovitz A, Kaur A, Urban E, Zehl M, Páchniková G, Wang Y, Kretschmer N, Slaninová I, Pauli GF, Franzblau SG, Krupitza G, Bauer R, Kopp B.
J Nat Prod (2014) 77 : 1069 -1073
PubMed 24725159 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 5.27 5.27

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL367881 (+)-USNIC ACID 1 5.27
CHEMBL173530 STICTIC ACID 1 -
CHEMBL3234666 1 -
CHEMBL229087 1 -
CHEMBL3234667 1 -
CHEMBL3234668 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL367881 (+)-USNIC ACID IC50 = 5400.0 nM 5.27
CHEMBL173530 STICTIC ACID IC50 > 10000.0 nM -
CHEMBL3234666 IC50 > 10000.0 nM -
CHEMBL229087 IC50 > 10000.0 nM -
CHEMBL3234667 IC50 > 10000.0 nM -
CHEMBL3234668 IC50 > 10000.0 nM -