Assay Detail
Binding
CHEMBL3266141
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to progesterone receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The discovery of potent and selective non-steroidal glucocorticoid receptor modulators, suitable for inhalation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.73 | 6.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3261407 | — | — | 1 | 6.11 |
| CHEMBL3261425 | — | — | 1 | 5.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3261407 | — | IC50 | = | 770.0 | nM | 6.11 |
| CHEMBL3261425 | — | IC50 | = | 4500.0 | nM | 5.35 |