Assay Detail
Functional
CHEMBL3266750
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at APJ receptor (unknown origin) expressed in CHO cells co-expressing with Calphaq16 assessed as calcium mobilization
33
Total Activities
33
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identifying structural determinants of potency for analogs of apelin-13: integration of C-terminal truncation with structure-activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 33 | 7.51 | 9.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3184840 | — | — | 1 | 9.38 |
| CHEMBL414173 | — | — | 1 | 9.06 |
| CHEMBL3261778 | — | — | 1 | 8.96 |
| CHEMBL3261787 | — | — | 1 | 8.77 |
| CHEMBL3261776 | — | — | 1 | 8.72 |
| CHEMBL3261789 | — | — | 1 | 8.66 |
| CHEMBL3261786 | — | — | 1 | 8.49 |
| CHEMBL3261773 | — | — | 1 | 8.36 |
| CHEMBL3261774 | — | — | 1 | 8.33 |
| CHEMBL3261780 | — | — | 1 | 8.05 |
| CHEMBL3261767 | — | — | 1 | 7.72 |
| CHEMBL3261766 | — | — | 1 | 7.70 |
| CHEMBL3261779 | — | — | 1 | 7.51 |
| CHEMBL3262012 | — | — | 1 | 7.48 |
| CHEMBL3261788 | — | — | 1 | 7.36 |
| CHEMBL3261790 | — | — | 1 | 7.14 |
| CHEMBL3262016 | — | — | 1 | 7.08 |
| CHEMBL3261783 | — | — | 1 | 6.62 |
| CHEMBL3261784 | — | — | 1 | 6.31 |
| CHEMBL3262011 | — | — | 1 | 6.27 |
| CHEMBL3261782 | — | — | 1 | 6.20 |
| CHEMBL3261775 | — | — | 1 | 6.16 |
| CHEMBL3261781 | — | — | 1 | 6.03 |
| CHEMBL3261777 | — | — | 1 | 5.86 |
| CHEMBL3261768 | — | — | 1 | 5.63 |
| CHEMBL3261769 | — | — | 1 | - |
| CHEMBL3261770 | — | — | 1 | - |
| CHEMBL3261771 | — | — | 1 | - |
| CHEMBL3261772 | — | — | 1 | - |
| CHEMBL3261785 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3184840 | — | EC50 | = | 0.42 | nM | 9.38 |
| CHEMBL414173 | — | EC50 | = | 0.87 | nM | 9.06 |
| CHEMBL3261778 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL3261787 | — | EC50 | = | 1.7 | nM | 8.77 |
| CHEMBL3261776 | — | EC50 | = | 1.9 | nM | 8.72 |
| CHEMBL3261789 | — | EC50 | = | 2.2 | nM | 8.66 |
| CHEMBL3261786 | — | EC50 | = | 3.2 | nM | 8.49 |
| CHEMBL3261773 | — | EC50 | = | 4.4 | nM | 8.36 |
| CHEMBL3261774 | — | EC50 | = | 4.7 | nM | 8.33 |
| CHEMBL3261780 | — | EC50 | = | 8.9 | nM | 8.05 |
| CHEMBL3261767 | — | EC50 | = | 19.0 | nM | 7.72 |
| CHEMBL3261766 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3261779 | — | EC50 | = | 31.0 | nM | 7.51 |
| CHEMBL3262012 | — | EC50 | = | 33.0 | nM | 7.48 |
| CHEMBL3261788 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL3261790 | — | EC50 | = | 73.0 | nM | 7.14 |
| CHEMBL3262016 | — | EC50 | = | 83.18 | nM | 7.08 |
| CHEMBL3261783 | — | EC50 | = | 237.0 | nM | 6.62 |
| CHEMBL3261784 | — | EC50 | = | 494.0 | nM | 6.31 |
| CHEMBL3262011 | — | EC50 | = | 539.0 | nM | 6.27 |
| CHEMBL3261782 | — | EC50 | = | 637.0 | nM | 6.20 |
| CHEMBL3261775 | — | EC50 | = | 691.0 | nM | 6.16 |
| CHEMBL3261781 | — | EC50 | = | 936.0 | nM | 6.03 |
| CHEMBL3261777 | — | EC50 | = | 1383.0 | nM | 5.86 |
| CHEMBL3261768 | — | EC50 | = | 2350.0 | nM | 5.63 |
| CHEMBL3261769 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3261770 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3261771 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3261772 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3261785 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3262013 | — | EC50 | > | 3000.0 | nM | - |
| CHEMBL3262015 | — | EC50 | > | 31622.78 | nM | - |
| CHEMBL3262014 | — | EC50 | > | 31622.78 | nM | - |