Assay Detail
Functional
CHEMBL3267829
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Inhibition of human HCT116 cell growth after 96 hrs by counting kit-8 analysis
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HCT-116 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Optimizing the Physicochemical Properties of Raf/MEK Inhibitors by Nitrogen Scanning.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 7.08 | 7.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3092195 | — | — | 1 | 7.77 |
| CHEMBL3092179 | — | — | 1 | 7.66 |
| CHEMBL3092189 | — | — | 1 | 7.62 |
| CHEMBL3263996 | — | — | 1 | 7.50 |
| CHEMBL3264002 | AVUTOMETINIB | 3.0 | 1 | 7.40 |
| CHEMBL3264000 | — | — | 1 | 7.35 |
| CHEMBL3263999 | — | — | 1 | 6.96 |
| CHEMBL3263995 | — | — | 1 | 6.57 |
| CHEMBL3264001 | — | — | 1 | 6.05 |
| CHEMBL3263994 | — | — | 1 | 5.96 |
| CHEMBL3263997 | — | — | 1 | - |
| CHEMBL3263998 | — | — | 1 | - |
| CHEMBL3264003 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3092195 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL3092179 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL3092189 | — | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL3263996 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL3264002 | AVUTOMETINIB | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL3264000 | — | IC50 | = | 45.0 | nM | 7.35 |
| CHEMBL3263999 | — | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL3263995 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL3264001 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL3263994 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL3263997 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3263998 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL3264003 | — | IC50 | > | 10000.0 | nM | - |