Assay Detail
Binding
CHEMBL3269019
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human SQS
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Multitarget drug discovery for tuberculosis and other infectious diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.00 | 4.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL561057 | SQ109 | 2.0 | 1 | 4.00 |
| CHEMBL3261880 | — | — | 1 | 4.00 |
| CHEMBL3261881 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL561057 | SQ109 | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL3261880 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL3261881 | — | IC50 | = | 100000.0 | nM | 4.00 |